Synthesis and biological activity of permethrinic acid analogs containing various substituents in position 2 of the cyclopropane ring

被引：10

作者：

Mirzabekova, N. S. ^{[1
]}

Kuz'mina, N. E. ^{[1
]}

Lukashov, O. I. ^{[1
]}

Sokolova, N. A. ^{[1
]}

Golosov, S. N. ^{[1
]}

Kazakov, P. V. ^{[1
]}

Perlova, T. G. ^{[2
]}

Potapova, V. V. ^{[2
]}

Kheinman, V. A. ^{[2
]}

Ivanova, G. B. ^{[2
]}

机构：

[1] State Res Inst Organ Chem & Technol, Moscow 111024, Russia

[2] All Russian Res Inst Chem Means Plant Protect, Moscow, Russia

来源：

RUSSIAN JOURNAL OF ORGANIC CHEMISTRY | 2008年 / 44卷 / 08期

关键词：

D O I：

10.1134/S107042800808006X

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A number of permethrinic acid ethyl ester derivatives having various substituents [Et, Pr, Ph, Ph(CH2)n (n = 1, 2), etc.] in position 2 of the cyclopropane ring were synthesized, and their insecticidal acivity against typhoid flies., rice weevils, and bean aphides, as well as juvenoid activity on flour beetle chrysalises, was studied. The newly synthesized Compounds turned out to exhibit weak insecticidal activity against standard insects but pronounced juvenile hormone activity, which differentiates them from permethrinic acid esters.

引用

页码：1139 / 1149

页数：11

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S. N. Golosov
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V. V. Potapova
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