Synthesis and biological activity of permethrinic acid analogs containing various substituents in position 2 of the cyclopropane ring

被引：10

作者：

Mirzabekova, N. S. ^{[1
]}

Kuz'mina, N. E. ^{[1
]}

Lukashov, O. I. ^{[1
]}

Sokolova, N. A. ^{[1
]}

Golosov, S. N. ^{[1
]}

Kazakov, P. V. ^{[1
]}

Perlova, T. G. ^{[2
]}

Potapova, V. V. ^{[2
]}

Kheinman, V. A. ^{[2
]}

Ivanova, G. B. ^{[2
]}

机构：

[1] State Res Inst Organ Chem & Technol, Moscow 111024, Russia

[2] All Russian Res Inst Chem Means Plant Protect, Moscow, Russia

来源：

RUSSIAN JOURNAL OF ORGANIC CHEMISTRY | 2008年 / 44卷 / 08期

关键词：

D O I：

10.1134/S107042800808006X

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A number of permethrinic acid ethyl ester derivatives having various substituents [Et, Pr, Ph, Ph(CH2)n (n = 1, 2), etc.] in position 2 of the cyclopropane ring were synthesized, and their insecticidal acivity against typhoid flies., rice weevils, and bean aphides, as well as juvenoid activity on flour beetle chrysalises, was studied. The newly synthesized Compounds turned out to exhibit weak insecticidal activity against standard insects but pronounced juvenile hormone activity, which differentiates them from permethrinic acid esters.

引用

页码：1139 / 1149

页数：11

共 50 条

[41] Quantitative structure-activity relationships of imidacloprid and its analogs with substituents at the C5 position on the pyridine ring in the neuroblocking activity
Nishimura, Keiichiro
Kiriyama, Kazuhisa
Kagabu, Shinzo
JOURNAL OF PESTICIDE SCIENCE, 2006, 31 (02) : 110 - 115
[42] STEROIDS .250. SYNTHESIS OF SOME 19-HYDROXYLATED ANDROGEN ANALOGS WITH THE CYCLOPROPANE RING IN 4,5-POSITION
JOSKA, J
FAJKOS, J
COLLECTION OF CZECHOSLOVAK CHEMICAL COMMUNICATIONS, 1981, 46 (11) : 2751 - 2757
[43] ON STEROIDS .272. SYNTHESIS OF 19-HYDROXYLATED ANALOGS OF ANDROSTENEDIONE AND TESTOSTERONE WITH THE CYCLOPROPANE RING IN 4,5-POSITION
JOSKA, J
FAJKOS, J
COLLECTION OF CZECHOSLOVAK CHEMICAL COMMUNICATIONS, 1982, 47 (09) : 2423 - 2432
[44] SYNTHESIS AND BIOLOGICAL-ACTIVITY OF ALLENIC ANALOGS OF ABSCISIC-ACID
ABRAMS, SR
MILBORROW, BV
PHYTOCHEMISTRY, 1991, 30 (10) : 3189 - 3195
[45] SYNTHESIS AND BIOLOGICAL-ACTIVITY OF STEROIDS CONTAINING A HETEROATOM IN RING-A
SHNER, VF
RULIN, VA
SUVOROV, NN
KHIMIKO-FARMATSEVTICHESKII ZHURNAL, 1978, 12 (04): : 22 - 37
[46] Synthesis and biological activity of conformationally defined retinoic acid analogs.
Atigadda, VR
Brouillette, WJ
Muccio, DD
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1999, 218 : U925 - U926
[47] Synthesis and biological activity of Tonghaosu analogs containing phenoxy-phenyl moiety
Chen, L
Xu, HH
Yin, BL
Xiao, C
Hu, TS
Wu, YL
CHINESE JOURNAL OF CHEMISTRY, 2004, 22 (09) : 984 - 989
[48] Synthesis and Biological Activity of Tonghaosu Analogs Containing Phenoxy-phenyl Moiety
陈立
徐汉虹
尹标林
肖春
胡泰山
吴毓林
Chinese Journal of Chemistry, 2004, (09) : 984 - 989
[49] Synthesis, structure, and biological activity of 4-hetaryl-2-pyrrolidones containing a pyrazole ring
Gorodnicheva, Natal'ya V.
Vasil'eva, Olga S.
Ostroglyadov, Evgeny S.
Baichurin, Ruslan I.
Litvinov, Igor A.
Tyurenkov, Ivan N.
Kovalev, Nikolay S.
Bakulin, Dmitry A.
Kurkin, Denis V.
Baichurina, Larisa V.
Makarenko, Sergey V.
CHEMISTRY OF HETEROCYCLIC COMPOUNDS, 2022, 58 (11) : 598 - 607
[50] Synthesis, structure, and biological activity of 4-hetaryl-2-pyrrolidones containing a pyrazole ring
Natal’ya V. Gorodnicheva
Olga S. Vasil’eva
Evgeny S. Ostroglyadov
Ruslan I. Baichurin
Igor A. Litvinov
Ivan N. Tyurenkov
Nikolay S. Kovalev
Dmitry A. Bakulin
Denis V. Kurkin
Larisa V. Baichurina
Sergey V. Makarenko
Chemistry of Heterocyclic Compounds, 2022, 58 : 598 - 607

← 1 2 3 4 5 →