Synthesis and biological activity of permethrinic acid analogs containing various substituents in position 2 of the cyclopropane ring

被引：0
|
作者：
N. S. Mirzabekova
N. E. Kuz’mina
O. I. Lukashov
N. A. Sokolova
S. N. Golosov
P. V. Kazakov
T. G. Perlova
V. V. Potapova
V. A. Kheinman
G. B. Ivanova
机构：
[1] State Research Institute of Organic Chemistry and Technology,
[2] All-Russian Research Institute of Chemical Means for Plant Protection,undefined
来源：
Russian Journal of Organic Chemistry | 2008年 / 44卷
关键词：
Chromatographic Purification; Cyclopropane Ring; Diethoxyphosphoryl; Rice Weevil; Graphic Purification;
D O I：
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中图分类号：
学科分类号：
摘要：
A number of permethrinic acid ethyl ester derivatives having various substituents [Et, Pr, Ph, Ph(CH2)n (n = 1, 2), etc.] in position 2 of the cyclopropane ring were synthesized, and their insecticidal acivity against typhoid flies, rice weevils, and bean aphides, as well as juvenoid activity on flour beetle chrysalises, was studied. The newly synthesized compounds turned out to exhibit weak insecticidal activity against standard insects but pronounced juvenile hormone activity, which differentiates them from permethrinic acid esters.
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页码：1139 / 1149
页数：10
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