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- [11] A new family of H3 receptor antagonists based on the natural product ConessineBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2008, 18 (04) : 1490 - 1494Santora, Vincent J.论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USACovel, Jonathan A.论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USAHayashi, Rena论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USAHofilena, Brian J.论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USAIbarra, Jason B.论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USAPulley, Michelle D.论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USAWeinhouse, Michael I.论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USASengupta, Dipanjan论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USADuffield, Jonathan J.论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USASemple, Graeme论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USAWebb, Robert R.论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USASage, Carleton论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USARen, Albert论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USAPereira, Guilherme论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USAKnudsen, Jens论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USAEdwards, Jeffrey E.论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Drug Metab & Pharmacokinet, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USASuarez, Marissa论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Discovery Biol, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USAFrazer, John论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Discovery Biol, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USAThomsen, William论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Discovery Biol, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USAHauser, Erin论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Discovery Biol, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USAWhelan, Kevin论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Discovery Biol, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USAGrottick, Andrew J.论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Discovery Biol, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA
- [12] Drug-drug interaction potential and clinical pharmacokinetics of enerisant, a novel potent and selective histamine H3 receptor antagonistXENOBIOTICA, 2021, 51 (07) : 786 - 795Terasaka, Shuichi论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Drug Metab & Pharmacokinet, Drug Safety & Pharmacokinet Labs, Res Headquarters, Saitama, Japan Taisho Pharmaceut Co Ltd, Drug Metab & Pharmacokinet, Drug Safety & Pharmacokinet Labs, Res Headquarters, Saitama, JapanHachiuma, Kenji论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Drug Metab & Pharmacokinet, Drug Safety & Pharmacokinet Labs, Res Headquarters, Saitama, Japan Taisho Pharmaceut Co Ltd, Drug Metab & Pharmacokinet, Drug Safety & Pharmacokinet Labs, Res Headquarters, Saitama, JapanMano, Yoko论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Dev Headquarters, Tokyo, Japan Taisho Pharmaceut Co Ltd, Drug Metab & Pharmacokinet, Drug Safety & Pharmacokinet Labs, Res Headquarters, Saitama, JapanOnishi, Koichi论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Dev Headquarters, Tokyo, Japan Taisho Pharmaceut Co Ltd, Drug Metab & Pharmacokinet, Drug Safety & Pharmacokinet Labs, Res Headquarters, Saitama, JapanKitajima, Iwao论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Dev Headquarters, Tokyo, Japan Taisho Pharmaceut Co Ltd, Drug Metab & Pharmacokinet, Drug Safety & Pharmacokinet Labs, Res Headquarters, Saitama, JapanNishino, Izumi论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Dev Headquarters, Tokyo, Japan Taisho Pharmaceut Co Ltd, Drug Metab & Pharmacokinet, Drug Safety & Pharmacokinet Labs, Res Headquarters, Saitama, JapanEndo, Hiromi论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Drug Metab & Pharmacokinet, Drug Safety & Pharmacokinet Labs, Res Headquarters, Saitama, Japan Taisho Pharmaceut Co Ltd, Drug Metab & Pharmacokinet, Drug Safety & Pharmacokinet Labs, Res Headquarters, Saitama, Japan
- [13] A-320436:: Potent human non-imidazole histamine H3 receptor antagonist.ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2003, 225 : U217 - U217Curtis, MP论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Abbott Pk, IL 60064 USADwight, W论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Abbott Pk, IL 60064 USAFox, GB论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Abbott Pk, IL 60064 USAEsbenshade, TA论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Abbott Pk, IL 60064 USAPan, JB论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Abbott Pk, IL 60064 USABennani, YL论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Abbott Pk, IL 60064 USAHancock, AA论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Abbott Pk, IL 60064 USAFaghih, R论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Abbott Pk, IL 60064 USA
- [14] Pharmacological and behavioral properties of A-349821, a selective and potent human histamine H3 receptor antagonistBIOCHEMICAL PHARMACOLOGY, 2004, 68 (05) : 933 - 945Esbenshade, TA论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept Neurosci Res, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USA Abbott Labs, Dept Neurosci Res, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USAFox, GB论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept Neurosci Res, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USA Abbott Labs, Dept Neurosci Res, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USAKrueger, KM论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept Neurosci Res, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USA Abbott Labs, Dept Neurosci Res, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USABaranowski, JL论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept Neurosci Res, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USA Abbott Labs, Dept Neurosci Res, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USAMiller, TR论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept Neurosci Res, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USA Abbott Labs, Dept Neurosci Res, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USAKang, CH论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept Neurosci Res, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USA Abbott Labs, Dept Neurosci Res, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USADenny, LI论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept Neurosci Res, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USA Abbott Labs, Dept Neurosci Res, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USAWitte, DG论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept Neurosci Res, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USA Abbott Labs, Dept Neurosci Res, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USAYao, BB论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept Neurosci Res, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USA Abbott Labs, Dept Neurosci Res, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USAPan, JB论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept Neurosci Res, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USA Abbott Labs, Dept Neurosci Res, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USAFaghih, R论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept Neurosci Res, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USA Abbott Labs, Dept Neurosci Res, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USABennani, YL论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept Neurosci Res, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USA Abbott Labs, Dept Neurosci Res, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USAWilliams, M论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept Neurosci Res, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USA Abbott Labs, Dept Neurosci Res, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USAHancock, AA论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept Neurosci Res, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USA Abbott Labs, Dept Neurosci Res, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USA
- [15] MEDI 394-Design and synthesis of novel, potent and selective H3 antagonists based on the natural product conessineABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2007, 234Covel, Jonathan A.论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USAHayashi, Rena论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USAHofilena, Brian论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USAIbarra, Jason论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USAPulley, Michelle论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USAWeinhouse, Michael论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USASengupta, Dipanjan论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USADuffield, Jonathan论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USASantora, Vincent J.论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USASemple, Graeme论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USAWebb, Robert R.论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USASuarez, Marissa论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USAFrazer, John论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USAThompson, William论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USAEdwards, Jeffrey论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USAHauser, Erin论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USAWhelan, Kevin论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USAGrottick, Andrew论文数: 0 引用数: 0 h-index: 0机构: Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA Arena Pharmaceut, Med Chem, San Diego, CA 92121 USA
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