ULTRASOUND-ASSISTED N-ARYLATION OF INDOLES WITHOUT ANY CATALYST

被引：5
|
作者：
Xu, Hui [1 ]
Lv, Lei [1 ]
Fan, Ling-ling [1 ]
He, Xiao-qiang [1 ]
机构：
[1] NW A&F Univ, Coll Sci, Lab Pharmaceut Synth, Yangling 712100, Peoples R China
来源：
HETEROCYCLES | 2008年 / 76卷 / 01期
关键词：
Ultrasound-Assisted Reaction; N-Arylindole; Catalyst-Free; Synthesis;
D O I：
10.3987/COM-07-S(N)1
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
An efficient method for the ultrasound-assisted N-arylation of indoles with haloarenes in an air atmosphere mediated by CS2CO3 without any catalyst is reported. N-arylindoles are obtained in moderate to good yields while indoles cross-coupling with activated aryl halides (X = F or Cl).
引用
收藏
页码：249 / 256
页数：8
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