Simple and convenient synthesis of (±)-bakuchiol

被引：10
|
作者：
Chen, Hongli [1 ]
Li, Yuanchao [1 ]
机构：
[1] Chinese Acad Sci, Shanghai Inst Mat Med, Shanghai 201203, Peoples R China
来源：
LETTERS IN ORGANIC CHEMISTRY | 2008年 / 5卷 / 06期
关键词：
(+/-)-bakuchiol; citral; 1,4-addition; Grignard reagent;
D O I：
10.2174/157017808785740499
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A simple and convenient synthesis of (+/-)-bakuchiol has been developed. The key intermediate was obtained in only one step from the easily available starting material, citral, by an 1,4-addition procedure. (+/-)-Bakuchiol was finally produced in 4 steps to give 50% overall yield.
引用
收藏
页码：467 / 469
页数：3
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