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- [31] Discovery of MK-1084, a low dose selective clinical stage KRAS G12C inhibitorMOLECULAR CANCER THERAPEUTICS, 2023, 22 (12)Maddess, Matthew L.论文数: 0 引用数: 0 h-index: 0Sloman, David L.论文数: 0 引用数: 0 h-index: 0Ma, Xiaoshen论文数: 0 引用数: 0 h-index: 0Palani, Anandan论文数: 0 引用数: 0 h-index: 0Stoeck, Alexander论文数: 0 引用数: 0 h-index: 0Sather, Aaron C.论文数: 0 引用数: 0 h-index: 0Solban, Nicolas论文数: 0 引用数: 0 h-index: 0Duggal, Ruchia论文数: 0 引用数: 0 h-index: 0Ballard, Jeanine论文数: 0 引用数: 0 h-index: 0Munsell, Erik V.论文数: 0 引用数: 0 h-index: 0Chen, Lin-Chi论文数: 0 引用数: 0 h-index: 0Han, Yongxin论文数: 0 引用数: 0 h-index: 0Miller, Richard论文数: 0 引用数: 0 h-index: 0Gathiaka, Symon论文数: 0 引用数: 0 h-index: 0Brynczka, Christopher论文数: 0 引用数: 0 h-index: 0Li, Hongming论文数: 0 引用数: 0 h-index: 0Yang, Ruojing论文数: 0 引用数: 0 h-index: 0Brynczka, Christopher论文数: 0 引用数: 0 h-index: 0Day, Phil论文数: 0 引用数: 0 h-index: 0
- [32] The FAK/SRC axis mediates resistance to KRAS G12C inhibitors and its blockade can overcome KRAS inhibitor resistanceCANCER RESEARCH, 2024, 84 (06)Shibata, Yuji论文数: 0 引用数: 0 h-index: 0Udagawa, Hibiki论文数: 0 引用数: 0 h-index: 0Nilsson, Monique B.论文数: 0 引用数: 0 h-index: 0Robichaux, Jacqulyne论文数: 0 引用数: 0 h-index: 0Galan-Cobo, Ana论文数: 0 引用数: 0 h-index: 0Negrao, Marcelo论文数: 0 引用数: 0 h-index: 0Molkentine, David P.论文数: 0 引用数: 0 h-index: 0He, Junqin论文数: 0 引用数: 0 h-index: 0Poteete, Alissa论文数: 0 引用数: 0 h-index: 0Qian, Yu论文数: 0 引用数: 0 h-index: 0Huang, Qian论文数: 0 引用数: 0 h-index: 0Skoulidis, Ferdinandos论文数: 0 引用数: 0 h-index: 0Heymach, John V.论文数: 0 引用数: 0 h-index: 0
- [33] Concomitant KRAS mutations attenuate sensitivity of non-small cell lung cancer cells to KRAS G12C inhibitionScientific Reports, 12Tereza Vaclova论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca,Translational Medicine, OncologyAtanu Chakraborty论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca,Translational Medicine, OncologyJames Sherwood论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca,Translational Medicine, OncologySarah Ross论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca,Translational Medicine, OncologyDanielle Carroll论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca,Translational Medicine, OncologyJ. Carl Barrett论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca,Translational Medicine, OncologyJulian Downward论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca,Translational Medicine, OncologyElza C. de Bruin论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca,Translational Medicine, Oncology
- [34] Quantifying KRAS G12C Covalent Drug Inhibitor Activity in Mouse Tumors Using Mass SpectrometryANALYTICAL CHEMISTRY, 2023, 95 (11) : 4834 - 4839Tran, John C.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Roche Grp, Biochem & Cellular Pharmacol, South San Francisco, CA 94080 USA Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USAHunsaker, Thomas论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USA Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USABell, Christina论文数: 0 引用数: 0 h-index: 0机构: CellCarta, Montreal, PQ H2X 3Y7, Canada Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USAMa, Taylur P.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Roche Grp, Microchem Prote & Lipid, South San Francisco, CA 94080 USA Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USAChan, Emily论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USA Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USALarrocha, Pablo Saenz-Lopez论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USA Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USAHomyk, Kelsey论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Roche Grp, Mol Oncol, South San Francisco, CA 94080 USA Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USALiu, Liling论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Roche Grp, Drug Metab & Pharmacokinet, South San Francisco, CA 94080 USA Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USALa, Hank论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Roche Grp, Drug Metab & Pharmacokinet, South San Francisco, CA 94080 USA Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USAMao, Jialin论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Roche Grp, Drug Metab & Pharmacokinet, South San Francisco, CA 94080 USA Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USAde la Cruz, Cecile C.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Roche Grp, Mol Oncol, South San Francisco, CA 94080 USA Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USAYu, Kebing论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Roche Grp, Microchem Prote & Lipid, South San Francisco, CA 94080 USA Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USABeresini, Maureen论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Roche Grp, Biochem & Cellular Pharmacol, South San Francisco, CA 94080 USA Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USAForrest, William F.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Roche Grp, OMNI Bioinformat, South San Francisco, CA 94080 USA Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USAXiao, Yang论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USA Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USAJang, Anne论文数: 0 引用数: 0 h-index: 0机构: CellCarta, Montreal, PQ H2X 3Y7, Canada Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USASamus, Natalia论文数: 0 引用数: 0 h-index: 0机构: CellCarta, Montreal, PQ H2X 3Y7, Canada Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USAStesco, Nicholas Dupuis论文数: 0 引用数: 0 h-index: 0机构: CellCarta, Montreal, PQ H2X 3Y7, Canada Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USAMentinova, Marija论文数: 0 引用数: 0 h-index: 0机构: CellCarta, Montreal, PQ H2X 3Y7, Canada Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USAParent, Stephane论文数: 0 引用数: 0 h-index: 0机构: CellCarta, Montreal, PQ H2X 3Y7, Canada Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USAPottiez, Gwenael论文数: 0 引用数: 0 h-index: 0机构: CellCarta, Montreal, PQ H2X 3Y7, Canada Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USASchirm, Michael论文数: 0 引用数: 0 h-index: 0机构: CellCarta, Montreal, PQ H2X 3Y7, Canada Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USAPurkey, Hans E.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Roche Grp, Discovery Chem, South San Francisco, CA 94080 USA Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USALiu, Yichin论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Roche Grp, Biochem & Cellular Pharmacol, South San Francisco, CA 94080 USA Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USAMerchant, Mark论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USA Genentech Inc, Translat Oncol, Roche Grp, South San Francisco, CA 94080 USA
- [35] Addressing Atropisomerism in the Development of Sotorasib, a Covalent Inhibitor of KRAS G12C: Structural, Analytical, and Synthetic ConsiderationsACCOUNTS OF CHEMICAL RESEARCH, 2022, 55 (20) : 2892 - 2903Lanman, Brian A.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Proc Dev, Drug Subst Technol, Cambridge, MA 02142 USAParsons, Andrew T.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Proc Dev, Drug Subst Technol, Cambridge, MA 02142 USA Amgen Inc, Dept Proc Dev, Drug Subst Technol, Cambridge, MA 02142 USAZech, Stephan G.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Lead Discovery & Characterizat, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Proc Dev, Drug Subst Technol, Cambridge, MA 02142 USA
- [36] Concomitant KRAS mutations attenuate sensitivity of non-small cell lung cancer cells to KRAS G12C inhibitionSCIENTIFIC REPORTS, 2022, 12 (01)Vaclova, Tereza论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Oncol, Translat Med, Cambridge CB4 0WG, England AstraZeneca, Oncol, Translat Med, Cambridge CB4 0WG, EnglandChakraborty, Atanu论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Oncol, Biosci, Cambridge CB2 0RE, England AstraZeneca, Oncol, Translat Med, Cambridge CB4 0WG, EnglandSherwood, James论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut, Precis Med & Biosamples, Cambridge CB4 0WG, England AstraZeneca, Oncol, Translat Med, Cambridge CB4 0WG, EnglandRoss, Sarah论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Oncol, Biosci, Cambridge CB2 0RE, England AstraZeneca, Oncol, Translat Med, Cambridge CB4 0WG, EnglandCarroll, Danielle论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Oncol, Translat Med, Cambridge CB4 0WG, England AstraZeneca, Oncol, Translat Med, Cambridge CB4 0WG, EnglandBarrett, J. Carl论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Oncol, Translat Med, Waltham, MA 02451 USA AstraZeneca, Oncol, Translat Med, Cambridge CB4 0WG, England论文数: 引用数: h-index:机构:de Bruin, Elza C.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Oncol, Translat Med, Cambridge CB4 0WG, England AstraZeneca, Oncol, Translat Med, Cambridge CB4 0WG, England
- [37] Characterisation of a novel KRAS G12C inhibitor ASP2453 that shows potent anti-tumour activity in KRAS G12C-mutated preclinical modelsBRITISH JOURNAL OF CANCER, 2022, 126 (05) : 744 - 753Nakayama, Ayako论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, Japan Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, JapanNagashima, Takeyuki论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, Japan Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, JapanNishizono, Yoshihiro论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, Japan Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, JapanKuramoto, Kazuyuki论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, Japan Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, JapanMori, Kenichi论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, Japan Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, JapanHomboh, Kazuya论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, Japan Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, JapanYuri, Masatoshi论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, Japan Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, JapanShimazaki, Masashi论文数: 0 引用数: 0 h-index: 0机构: Astellas Res Inst Amer LLC, Northbrook, IL USA Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, Japan
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- [40] Structure- based drug discovery of a selective, covalent KRas G12C inhibitor with oral activity in animal models of cancerABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2018, 256Fischer, John论文数: 0 引用数: 0 h-index: 0机构: Array Biopharma Inc, Boulder, CO USA Array Biopharma Inc, Boulder, CO USABaer, Brian论文数: 0 引用数: 0 h-index: 0机构: Array Biopharma Inc, Boulder, CO USA Array Biopharma Inc, Boulder, CO USABallard, Joshua论文数: 0 引用数: 0 h-index: 0机构: Array Biopharma Inc, Boulder, CO USA Array Biopharma Inc, Boulder, CO USABlake, James论文数: 0 引用数: 0 h-index: 0机构: Array Biopharma Inc, Boulder, CO USA Array Biopharma Inc, Boulder, CO USABouhana, Karyn论文数: 0 引用数: 0 h-index: 0机构: Array Biopharma Inc, Boulder, CO USA Array Biopharma Inc, Boulder, CO USABrandhuber, Barbara论文数: 0 引用数: 0 h-index: 0机构: Array Biopharma Inc, Boulder, CO USA Array Biopharma Inc, Boulder, CO USABriere, David论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA USA Array Biopharma Inc, Boulder, CO USABurgess, Laurence论文数: 0 引用数: 0 h-index: 0机构: Array Biopharma Inc, Boulder, CO USA Array Biopharma Inc, Boulder, CO USABurkard, Michael论文数: 0 引用数: 0 h-index: 0机构: Array Biopharma Inc, Boulder, CO USA Array Biopharma Inc, Boulder, CO USAChiang, Harrah论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA USA Array Biopharma Inc, Boulder, CO USAChicarelli, Mark论文数: 0 引用数: 0 h-index: 0机构: Array Biopharma Inc, Boulder, CO USA Array Biopharma Inc, Boulder, CO USAChristensen, James论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA USA Array Biopharma Inc, Boulder, CO USADavidson, Kevin论文数: 0 引用数: 0 h-index: 0机构: Array Biopharma Inc, Boulder, CO USA Array Biopharma Inc, Boulder, CO USAGaudino, John论文数: 0 引用数: 0 h-index: 0机构: Array Biopharma Inc, Boulder, CO USA Array Biopharma Inc, Boulder, CO USAHallin, Jill论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA USA Array Biopharma Inc, Boulder, CO USAHanson, Lauren论文数: 0 引用数: 0 h-index: 0机构: Array Biopharma Inc, Boulder, CO USA Array Biopharma Inc, Boulder, CO USAHee, Kenneth论文数: 0 引用数: 0 h-index: 0机构: Array Biopharma Inc, Boulder, CO USA Array Biopharma Inc, Boulder, CO USAHicken, Erik论文数: 0 引用数: 0 h-index: 0机构: Array Biopharma Inc, Boulder, CO USA Array Biopharma Inc, Boulder, CO USAHinklin, Ronald论文数: 0 引用数: 0 h-index: 0机构: Array Biopharma Inc, Boulder, CO USA Array Biopharma Inc, Boulder, CO USAMarx, Matthew论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA USA Array Biopharma Inc, Boulder, CO USAMejia, Macedonio论文数: 0 引用数: 0 h-index: 0机构: Array Biopharma Inc, Boulder, CO USA Array Biopharma Inc, Boulder, CO USAOlson, Peter论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA USA Array Biopharma Inc, Boulder, CO USASavechenkov, Pavel论文数: 0 引用数: 0 h-index: 0机构: Array Biopharma Inc, Boulder, CO USA Array Biopharma Inc, Boulder, CO USASudhakar, Niranjan论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA USA Array Biopharma Inc, Boulder, CO USATang, Tony论文数: 0 引用数: 0 h-index: 0机构: Array Biopharma Inc, Boulder, CO USA Array Biopharma Inc, Boulder, CO USAVigers, Guy论文数: 0 引用数: 0 h-index: 0机构: Array Biopharma Inc, Boulder, CO USA Array Biopharma Inc, Boulder, CO USAZecca, Henry论文数: 0 引用数: 0 h-index: 0机构: Array Biopharma Inc, Boulder, CO USA Array Biopharma Inc, Boulder, CO USAFell, Jay论文数: 0 引用数: 0 h-index: 0机构: Array Biopharma Inc, Boulder, CO USA Array Biopharma Inc, Boulder, CO USA