共 50 条
- [31] Discovery of a Novel p38α-MK2 Complex Inhibitor as a Potential Choice for Autoimmune DiseasesJOURNAL OF MEDICINAL CHEMISTRY, 2025, 68 (02) : 1328 - 1343Fu, Donglin论文数: 0 引用数: 0 h-index: 0机构: Changchun GeneSci Pharmaceut Co Ltd, Chem Pharmaceut Res Ctr, Shanghai 200120, Peoples R China Changchun GeneSci Pharmaceut Co Ltd, Chem Pharmaceut Res Ctr, Shanghai 200120, Peoples R ChinaYang, Zimo论文数: 0 引用数: 0 h-index: 0机构: Changchun GeneSci Pharmaceut Co Ltd, Chem Pharmaceut Res Ctr, Shanghai 200120, Peoples R China Changchun GeneSci Pharmaceut Co Ltd, Chem Pharmaceut Res Ctr, Shanghai 200120, Peoples R ChinaJia, Xiangyu论文数: 0 引用数: 0 h-index: 0机构: Changchun GeneSci Pharmaceut Co Ltd, Chem Pharmaceut Res Ctr, Shanghai 200120, Peoples R China Changchun GeneSci Pharmaceut Co Ltd, Chem Pharmaceut Res Ctr, Shanghai 200120, Peoples R ChinaHan, Tian论文数: 0 引用数: 0 h-index: 0机构: Changchun GeneSci Pharmaceut Co Ltd, Chem Pharmaceut Res Ctr, Shanghai 200120, Peoples R China Changchun GeneSci Pharmaceut Co Ltd, Chem Pharmaceut Res Ctr, Shanghai 200120, Peoples R ChinaHan, Long论文数: 0 引用数: 0 h-index: 0机构: Changchun GeneSci Pharmaceut Co Ltd, Chem Pharmaceut Res Ctr, Shanghai 200120, Peoples R China Changchun GeneSci Pharmaceut Co Ltd, Chem Pharmaceut Res Ctr, Shanghai 200120, Peoples R ChinaZhang, Xiaobing论文数: 0 引用数: 0 h-index: 0机构: Changchun GeneSci Pharmaceut Co Ltd, Chem Pharmaceut Res Ctr, Shanghai 200120, Peoples R China Changchun GeneSci Pharmaceut Co Ltd, Chem Pharmaceut Res Ctr, Shanghai 200120, Peoples R ChinaXia, Yuanfeng论文数: 0 引用数: 0 h-index: 0机构: Changchun GeneSci Pharmaceut Co Ltd, Chem Pharmaceut Res Ctr, Shanghai 200120, Peoples R China Changchun GeneSci Pharmaceut Co Ltd, Chem Pharmaceut Res Ctr, Shanghai 200120, Peoples R ChinaWang, Siqin论文数: 0 引用数: 0 h-index: 0机构: Changchun GeneSci Pharmaceut Co Ltd, Shanghai 200120, Peoples R China Changchun GeneSci Pharmaceut Co Ltd, Chem Pharmaceut Res Ctr, Shanghai 200120, Peoples R ChinaJin, Lei论文数: 0 引用数: 0 h-index: 0机构: Changchun GeneSci Pharmaceut Co Ltd, Shanghai 200120, Peoples R China Changchun GeneSci Pharmaceut Co Ltd, Chem Pharmaceut Res Ctr, Shanghai 200120, Peoples R ChinaHu, Zhilong论文数: 0 引用数: 0 h-index: 0机构: Changchun GeneSci Pharmaceut Co Ltd, Chem Pharmaceut Res Ctr, Shanghai 200120, Peoples R China Changchun GeneSci Pharmaceut Co Ltd, Chem Pharmaceut Res Ctr, Shanghai 200120, Peoples R ChinaYang, Fanglong论文数: 0 引用数: 0 h-index: 0机构: Changchun GeneSci Pharmaceut Co Ltd, Chem Pharmaceut Res Ctr, Shanghai 200120, Peoples R China Changchun GeneSci Pharmaceut Co Ltd, Chem Pharmaceut Res Ctr, Shanghai 200120, Peoples R China
- [32] Rilonacept -: IL-1 inhibitor treatment of autoimmune diseases treatment of inflammatoty disordersDRUGS OF THE FUTURE, 2007, 32 (05) : 411 - 416Sorbera, L. A.论文数: 0 引用数: 0 h-index: 0机构: Univ Politecn Cataluna, E-08080 Barcelona, Spain Univ Politecn Cataluna, E-08080 Barcelona, SpainBozzo, J.论文数: 0 引用数: 0 h-index: 0机构: Univ Politecn Cataluna, E-08080 Barcelona, Spain Univ Politecn Cataluna, E-08080 Barcelona, SpainBayes, M.论文数: 0 引用数: 0 h-index: 0机构: Univ Politecn Cataluna, E-08080 Barcelona, Spain Univ Politecn Cataluna, E-08080 Barcelona, Spain
- [33] Discovery of Clinical Candidate GLPG3970: A Potent and Selective Dual SIK2/SIK3 Inhibitor for the Treatment of Autoimmune and Inflammatory DiseasesJOURNAL OF MEDICINAL CHEMISTRY, 2024, 67 (07) : 5233 - 5258Peixoto, Christophe论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceJoncour, Agnes论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceTemal-Laib, Taoues论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceTirera, Amynata论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceDos Santos, Aurelie论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceJary, Helene论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceBucher, Denis论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceLaenen, Wendy论文数: 0 引用数: 0 h-index: 0机构: Galapagos NV, B-2800 Mechelen, Belgium Galapagos SASU, F-93230 Romainville, FranceFernandes, Anna Pereira论文数: 0 引用数: 0 h-index: 0机构: Galapagos NV, B-2800 Mechelen, Belgium Galapagos SASU, F-93230 Romainville, FranceLavazais, Stephanie论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceDelachaume, Carole论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceMerciris, Didier论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceSaccomani, Corinne论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceDrennan, Michael论文数: 0 引用数: 0 h-index: 0机构: Galapagos NV, B-2800 Mechelen, Belgium Galapagos SASU, F-93230 Romainville, FranceLopez-Ramos, Miriam论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceWakselman, Emanuelle论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceDupont, Sonia论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceBorgonovi, Monica论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceMagadan, Carlos Roca论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceMonjardet, Alain论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceBrys, Reginald论文数: 0 引用数: 0 h-index: 0机构: Galapagos NV, B-2800 Mechelen, Belgium Galapagos SASU, F-93230 Romainville, FranceDe Vos, Steve论文数: 0 引用数: 0 h-index: 0机构: Galapagos NV, B-2800 Mechelen, Belgium Galapagos SASU, F-93230 Romainville, FranceAndrews, Martin论文数: 0 引用数: 0 h-index: 0机构: Galapagos NV, B-2800 Mechelen, Belgium Galapagos SASU, F-93230 Romainville, FranceJimenez, Juan-Miguel论文数: 0 引用数: 0 h-index: 0机构: Galapagos NV, B-2800 Mechelen, Belgium Galapagos SASU, F-93230 Romainville, FranceAmantini, David论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceDesroy, Nicolas论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, France
- [34] Discovery of CP-690,550: A Potent and Selective Janus Kinase (JAK) Inhibitor for the Treatment of Autoimmune Diseases and Organ Transplant RejectionJOURNAL OF MEDICINAL CHEMISTRY, 2010, 53 (24) : 8468 - 8484Flanagan, Mark E.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USABlumenkopf, Todd A.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, New London, CT 06320 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USABrissette, William H.论文数: 0 引用数: 0 h-index: 0机构: Yale Univ, New Haven, CT 06520 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USABrown, Matthew F.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USACasavant, Jeffrey M.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USAShang-Poa, Chang论文数: 0 引用数: 0 h-index: 0机构: Univ Connecticut, Dept Stat, Storrs, CT 06269 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USADoty, Jonathan L.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USAElliott, Eileen A.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USAFisher, Michael B.论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Ridgefield, CT 06877 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USAHines, Michael论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USAKent, Craig论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USAKudlacz, Elizabeth M.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, New London, CT 06320 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USALillie, Brett M.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USAMagnuson, Kelly S.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, New London, CT 06320 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USAMcCurdy, Sandra P.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USAMunchhof, Michael J.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USAPerry, Bret D.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USASawyer, Perry S.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USAStrelevitz, Timothy J.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USASubramanyam, Chakrapani论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USASun, Jianmin论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USAWhipple, David A.论文数: 0 引用数: 0 h-index: 0机构: Univ Kansas, Del Shankel Struct Biol Ctr, Lawrence, KS 66047 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USAChangelian, Paul S.论文数: 0 引用数: 0 h-index: 0机构: Lycera Corp, Plymouth, MI 48170 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA
- [35] First-in-class inhibitor of the T cell receptor for the treatment of autoimmune diseasesSCIENCE TRANSLATIONAL MEDICINE, 2016, 8 (370)论文数: 引用数: h-index:机构:Reyes-Garau, Diana论文数: 0 引用数: 0 h-index: 0机构: Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, SpainJimenez, M. Angeles论文数: 0 引用数: 0 h-index: 0机构: CSIC, Inst Quim Fis Rocasolano, Madrid, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, SpainCarrasco, Esther论文数: 0 引用数: 0 h-index: 0机构: Inst Adv Chem Catalonia IQAC CSIC, Barcelona, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, SpainMoreno, Beatriz论文数: 0 引用数: 0 h-index: 0机构: Hosp Clin Barcelona, Inst Invest Biomed August Pi i Sunyer, Barcelona, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, SpainMartinez-Pasamar, Sara论文数: 0 引用数: 0 h-index: 0机构: Hosp Clin Barcelona, Inst Invest Biomed August Pi i Sunyer, Barcelona, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, SpainCortes, Jose R.论文数: 0 引用数: 0 h-index: 0机构: Fdn Ctr Nacl Invest Cardiovasc Carlos III CNIC, Madrid, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, SpainPerona, Almudena论文数: 0 引用数: 0 h-index: 0机构: Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, Spain UAM, SmartLigs Bioinformat SL, Fdn Parque Cient Madrid, Campus Cantoblanco, Madrid, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, SpainAbia, David论文数: 0 引用数: 0 h-index: 0机构: Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, SpainBlanco, Soledad论文数: 0 引用数: 0 h-index: 0机构: Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, SpainFuentes, Manuel论文数: 0 引用数: 0 h-index: 0机构: Univ Salamanca, CSIC, Inst Invest Biomed Salamanca IBSAL, Ctr Invest Canc, Salamanca, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, SpainArellano, Irene论文数: 0 引用数: 0 h-index: 0机构: Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, SpainLobo, Juan论文数: 0 引用数: 0 h-index: 0机构: Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, SpainHeidarieh, Haleh论文数: 0 引用数: 0 h-index: 0机构: Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, SpainRueda, Javier论文数: 0 引用数: 0 h-index: 0机构: Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, Spain论文数: 引用数: h-index:机构:Cibrian, Danay论文数: 0 引用数: 0 h-index: 0机构: Fdn Ctr Nacl Invest Cardiovasc Carlos III CNIC, Madrid, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, SpainMartinez-Riano, Ana论文数: 0 引用数: 0 h-index: 0机构: Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, SpainMendoza, Pilar论文数: 0 引用数: 0 h-index: 0机构: Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, SpainPrieto, Cristina论文数: 0 引用数: 0 h-index: 0机构: Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, SpainCalleja, Enrique论文数: 0 引用数: 0 h-index: 0机构: Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, Spain论文数: 引用数: h-index:机构:Orfao, Alberto论文数: 0 引用数: 0 h-index: 0机构: Univ Salamanca, CSIC, Inst Invest Biomed Salamanca IBSAL, Ctr Invest Canc, Salamanca, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, SpainFresno, Manuel论文数: 0 引用数: 0 h-index: 0机构: Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, SpainSanchez-Madrid, Francisco论文数: 0 引用数: 0 h-index: 0机构: Fdn Ctr Nacl Invest Cardiovasc Carlos III CNIC, Madrid, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, SpainAlcami, Antonio论文数: 0 引用数: 0 h-index: 0机构: Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, SpainBovolenta, Paola论文数: 0 引用数: 0 h-index: 0机构: Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, SpainMartin, Pilar论文数: 0 引用数: 0 h-index: 0机构: Fdn Ctr Nacl Invest Cardiovasc Carlos III CNIC, Madrid, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, SpainVilloslada, Pablo论文数: 0 引用数: 0 h-index: 0机构: Hosp Clin Barcelona, Inst Invest Biomed August Pi i Sunyer, Barcelona, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, SpainMorreale, Antonio论文数: 0 引用数: 0 h-index: 0机构: Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, SpainMesseguer, Angel论文数: 0 引用数: 0 h-index: 0机构: Inst Adv Chem Catalonia IQAC CSIC, Barcelona, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, SpainAlarcon, Balbino论文数: 0 引用数: 0 h-index: 0机构: Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, Spain Autonomous Univ Madrid, CSIC UAM, Spanish Natl Res Council, Ctr Biol Mol Severo Ochoa, Madrid, Spain
- [36] Apremilast: a novel PDE4 inhibitor in the treatment of autoimmune and inflammatory diseasesTHERAPEUTIC ADVANCES IN MUSCULOSKELETAL DISEASE, 2010, 2 (05) : 271 - 278Schett, Georg论文数: 0 引用数: 0 h-index: 0机构: Univ Erlangen Nurnberg, Dept Internal Med 3, Rheumatol & Immunol, Krankenhausstr 12, D-91054 Erlangen, Germany Univ Erlangen Nurnberg, Dept Internal Med 3, Rheumatol & Immunol, Krankenhausstr 12, D-91054 Erlangen, GermanySloan, Victor S.论文数: 0 引用数: 0 h-index: 0机构: Celgene Corp, Summit, NJ USA Univ Erlangen Nurnberg, Dept Internal Med 3, Rheumatol & Immunol, Krankenhausstr 12, D-91054 Erlangen, GermanyStevens, Randall M.论文数: 0 引用数: 0 h-index: 0机构: Celgene Corp, Summit, NJ USA Univ Erlangen Nurnberg, Dept Internal Med 3, Rheumatol & Immunol, Krankenhausstr 12, D-91054 Erlangen, GermanySchafer, Peter论文数: 0 引用数: 0 h-index: 0机构: Celgene Corp, Summit, NJ USA Univ Erlangen Nurnberg, Dept Internal Med 3, Rheumatol & Immunol, Krankenhausstr 12, D-91054 Erlangen, Germany
- [37] Discovery of a new cytosolic phospholipase A2 inhibitor as a promising drug candidate for treatment of respiratory diseasesJOURNAL OF PHARMACOLOGICAL SCIENCES, 2016, 130 (03) : S73 - S73Terakawa, Maki论文数: 0 引用数: 0 h-index: 0机构: Asubio Pharma Co Ltd, Kobe, Hyogo, Japan Asubio Pharma Co Ltd, Kobe, Hyogo, JapanTomoo, Toshiyuki论文数: 0 引用数: 0 h-index: 0机构: Asubio Pharma Co Ltd, Kobe, Hyogo, Japan Asubio Pharma Co Ltd, Kobe, Hyogo, JapanHayashi, Yasuhiro论文数: 0 引用数: 0 h-index: 0机构: Asubio Pharma Co Ltd, Kobe, Hyogo, Japan Asubio Pharma Co Ltd, Kobe, Hyogo, JapanNagahira, Kazuhiro论文数: 0 引用数: 0 h-index: 0机构: Asubio Pharma Co Ltd, Kobe, Hyogo, Japan Asubio Pharma Co Ltd, Kobe, Hyogo, Japan
- [38] Autoimmune Rheumatic Diseases 2 Systemic lupus erythematosus and other autoimmune rheumatic diseases: challenges to treatmentLANCET, 2013, 382 (9894): : 809 - 818Murphy, Grainne论文数: 0 引用数: 0 h-index: 0机构: Univ Coll London Hosp, Ctr Rheumatol, Dept Med, London WC1E 6JF, England Univ Coll London Hosp, Ctr Rheumatol, Dept Med, London WC1E 6JF, EnglandLisnevskaia, Larissa论文数: 0 引用数: 0 h-index: 0机构: Oshawa Clin, Oshawa, ON, Canada Univ Coll London Hosp, Ctr Rheumatol, Dept Med, London WC1E 6JF, EnglandIsenberg, David论文数: 0 引用数: 0 h-index: 0机构: Univ Coll London Hosp, Ctr Rheumatol, Dept Med, London WC1E 6JF, England Univ Coll London Hosp, Ctr Rheumatol, Dept Med, London WC1E 6JF, England
- [39] Discovery of a potent and selective c-Kit inhibitor for the treatment of inflammatory diseasesBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2008, 18 (14) : 4137 - 4141Chen, Ning论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USABurli, Roland W.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USANeira, Susana论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAHungate, Randall论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAZhang, Dawei论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAYu, Violeta论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept HTS & Mol Pharmacol, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USANguyen, Yen论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept HTS & Mol Pharmacol, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USATudor, Yanyan论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept HTS & Mol Pharmacol, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAPlant, Matthew论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Inflammat, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAFlynn, Shaun论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept HTS & Mol Pharmacol, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAMeagher, Kristin L.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Mol Struct, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USALee, Matthew R.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Mol Struct, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAZhang, Xuxia论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Inflammat, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAItano, Andrea论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Inflammat, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USASchrag, Michael论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmacokinet & Drug Metab, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAXu, Yang论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmacokinet & Drug Metab, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USANg, Gordon Y.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Inflammat, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAHu, Essa论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USA
- [40] Discovery of a dual CCR2/CCR5 antagonist with a superior cardiovascular profile for the treatment of autoimmune diseasesABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2011, 242Hughes, Robert O.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Res & Dev, Cambridge, MA 02451 USA Pfizer Res & Dev, Cambridge, MA 02451 USARogier, D. Joseph论文数: 0 引用数: 0 h-index: 0机构: Pfizer Res & Dev, Cambridge, MA 02451 USA Pfizer Res & Dev, Cambridge, MA 02451 USADevraj, Rajesh论文数: 0 引用数: 0 h-index: 0机构: Pfizer Res & Dev, Cambridge, MA 02451 USA Pfizer Res & Dev, Cambridge, MA 02451 USAXue, Chu-Biao论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Willmington, DE 19880 USA Pfizer Res & Dev, Cambridge, MA 02451 USACao, Ganfeng论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Willmington, DE 19880 USA Pfizer Res & Dev, Cambridge, MA 02451 USATurner, Steven R.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Res & Dev, Cambridge, MA 02451 USA Pfizer Res & Dev, Cambridge, MA 02451 USAMorton, Philip A.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Res & Dev, Cambridge, MA 02451 USA Pfizer Res & Dev, Cambridge, MA 02451 USAKeys, Kelly论文数: 0 引用数: 0 h-index: 0机构: Pfizer Res & Dev, Cambridge, MA 02451 USA Pfizer Res & Dev, Cambridge, MA 02451 USACovington, Maryanne论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Willmington, DE 19880 USA Pfizer Res & Dev, Cambridge, MA 02451 USABond, Brian R.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Res & Dev, Cambridge, MA 02451 USA Pfizer Res & Dev, Cambridge, MA 02451 USAYu, Ying论文数: 0 引用数: 0 h-index: 0机构: Pfizer Res & Dev, Cambridge, MA 02451 USA Pfizer Res & Dev, Cambridge, MA 02451 USAMeade, Holly论文数: 0 引用数: 0 h-index: 0机构: Pfizer Res & Dev, Cambridge, MA 02451 USA Pfizer Res & Dev, Cambridge, MA 02451 USAHood, William F.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Res & Dev, Cambridge, MA 02451 USA Pfizer Res & Dev, Cambridge, MA 02451 USARoeberds, Steve论文数: 0 引用数: 0 h-index: 0机构: Pfizer Res & Dev, Cambridge, MA 02451 USA Pfizer Res & Dev, Cambridge, MA 02451 USANewton, Robert论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Willmington, DE 19880 USA Pfizer Res & Dev, Cambridge, MA 02451 USAMetcalf, Brian论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Willmington, DE 19880 USA Pfizer Res & Dev, Cambridge, MA 02451 USA