TY-0584: A potent, orally available small molecule YAP/TEAD inhibitor, exhibits anti-tumor effects in vitro and in vivo

被引:3
|
作者
Liang, Apeng
Dong, Shengli
Liu, Guangbin
Guo, Zhengfei
Li, Meihua
Han, Shuaibo
Cao, Yundi
Tu, Yian
Zhou, Chao
Yu, Yu
Xiao, Linglin
Huang, Wei
Yang, Xinlong
Fang, Lian
Li, Haoyun
Niu, Chengshan
Jiang, Mingyu
Xing, Feng
Chen, Shaoqing
Li, Jun
Wu, Yusheng
机构
关键词
D O I
10.1158/1538-7445.AM2023-4491
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
4491
引用
收藏
页数:3
相关论文
共 50 条
  • [41] KRC-108 as a Potent C-Met/Ron/Flt3 Kinase Inhibitor with Anti-tumor Effects in Vitro and in Vivo
    Han, S. Y.
    Kong, J. Y.
    Woo, D. K.
    Chin, Y. W.
    Cho, S. Y.
    Ha, J. D.
    Kim, H. R.
    Jeong, Y. J.
    Lee, J.
    EUROPEAN JOURNAL OF CANCER, 2012, 48 : S226 - S227
  • [42] Highly potent, orally active novel small-molecule HPK1 inhibitor DS21150768 induces anti-tumor responses in multiple syngeneic tumor mouse models
    Setsu, Genzui
    Goto, Megumi
    Ito, Kentaro
    Taira, Tomoe
    Miyamoto, Masaya
    Watanabe, Tomohiro
    Taniguchi, Toru
    Umezaki, Yuma
    Nakazawa, Yusuke
    Uesugi, Shuhei
    Mori, Kazuki
    Horiuchi, Takao
    Obuchi, Wataru
    Minami, Masako
    Shimada, Takashi
    Wada, Chisa
    Yoshida, Takanori
    Higuchi, Saito
    EUROPEAN JOURNAL OF PHARMACOLOGY, 2023, 961
  • [43] Anti-tumor effects of a small molecule C-C chemokine receptor 4 inhibitor in mouse tumor models
    Li, C.
    Campbell, J. J.
    Ertl, L. S.
    Miao, Z.
    Chhina, V.
    Kumamoto, A.
    Yau, S.
    Dang, T.
    Zhang, P.
    Schall, T. J.
    Singh, R.
    ANNALS OF ONCOLOGY, 2018, 29
  • [44] In vitro and in vivo Anti-Tumor Effects of Pan-HER Inhibitor Varlitinib on Cholangiocarcinoma Cell Lines
    Dokduang, Hasaya
    Jamnongkarn, Wassana
    Promraksa, Bundit
    Suksawat, Manida
    Padthaisong, Sureerat
    Thanee, Malinee
    Phetcharaburanin, Jutarop
    Namwat, Nisana
    Sangkhamanon, Sakkarn
    Titapun, Attapol
    Khuntikeo, Narong
    Klanrit, Poramate
    Loilome, Watcharin
    DRUG DESIGN DEVELOPMENT AND THERAPY, 2020, 14 : 2319 - 2334
  • [45] A novel cyclic peptide inhibitor targeting the YAP-TEAD protein-protein interaction shows potent anti-tumor effect in a variety of human malignancies including mesothelioma
    Hu, Yi P.
    Wang, Yinghua M.
    Lee, Daniel
    Ren, Yi
    CANCER RESEARCH, 2020, 80 (16)
  • [46] RAD140, an orally available selective androgen receptor modulator, exhibits potent anti-tumor activity in ER plus AR plus breast cancer models
    Yu, Z.
    Brown, J.
    Saeh, J.
    Hattersley, G.
    EUROPEAN JOURNAL OF CANCER, 2016, 69 : S149 - S149
  • [47] Rogaratinib, a small molecule pan-FGFR inhibitor potently inhibits FGFR4-phosphorylation and exerts anti-tumor efficacy in vivo and in vitro
    Politz, Oliver
    Gruenewald, Sylvia
    Walter, Alexander
    Siegel, Franziska
    Scholz, Arne
    Bender, Sebastian
    Kneip, Christoph
    Ellinghaus, Peter
    CANCER RESEARCH, 2018, 78 (13)
  • [48] In vitro and in vivo antitumor activities of T-3764518, a novel and orally available small molecule stearoyl-CoA desaturase 1 inhibitor
    Nishizawa, Satoru
    Sumi, Hiroyuki
    Satoh, Yoshihiko
    Yamamoto, Yukiko
    Kitazawa, Satoshi
    Honda, Kohei
    Araki, Hideo
    Kakoi, Kazuyo
    Imamura, Keisuke
    Sasaki, Masako
    Miyahisa, Ikuo
    Satomi, Yoshinori
    Nishigaki, Ryuuichi
    Hirayama, Megumi
    Aoyama, Kazunobu
    Maezaki, Hironobu
    Hara, Takahito
    EUROPEAN JOURNAL OF PHARMACOLOGY, 2017, 807 : 21 - 31
  • [49] Isoliquiritigenin, an Orally Available Natural FLT3 Inhibitor from Licorice, Exhibits Selective Anti-Acute Myeloid Leukemia Efficacy In Vitro and In Vivo
    Cao, Zhi-Xing
    Wen, Yi
    He, Jun-Lin
    Huang, Shen-Zhen
    Gao, Fei
    Guo, Chuan-Jie
    Liu, Qing-Qing
    Zheng, Shu-Wen
    Gong, Dao-Yin
    Li, Yu-Zhi
    Zhang, Ruo-Qi
    Chen, Jian-Ping
    Peng, Cheng
    MOLECULAR PHARMACOLOGY, 2019, 96 (05) : 589 - 599
  • [50] B13, a well-tolerated inhibitor of hedgehog pathway, exhibited potent anti-tumor effects against colorectal carcinoma in vitro and in vivo
    Wu, Huanxian
    Zhang, Lishun
    Chen, Boyu
    Ou, Baofang
    Xu, Jiahuan
    Tian, Nannan
    Yang, Danni
    Ai, Yangcheng
    Chen, Qianqing
    Quan, Dongling
    Zhang, Tingting
    Lv, Lin
    Tian, Yuanxin
    Zhang, Jiajie
    Wu, Shaoyu
    BIOORGANIC CHEMISTRY, 2023, 135