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- [1] Potent small molecule TEAD inhibitors targeting the Hippo pathway exhibit antiproliferation in vitro and anti-tumor effect in vivoCANCER RESEARCH, 2020, 80 (16)Amidon, Ben论文数: 0 引用数: 0 h-index: 0机构: Ikena Oncol, Boston, MA USA Ikena Oncol, Boston, MA USASyed, Sakeena论文数: 0 引用数: 0 h-index: 0机构: Ikena Oncol, Boston, MA USA Ikena Oncol, Boston, MA USACavanaugh, Jill论文数: 0 引用数: 0 h-index: 0机构: Ikena Oncol, Boston, MA USA Ikena Oncol, Boston, MA USAFrosch, Hyejin论文数: 0 引用数: 0 h-index: 0机构: Ikena Oncol, Boston, MA USA Ikena Oncol, Boston, MA USANatarajan, Prabitha论文数: 0 引用数: 0 h-index: 0机构: Ikena Oncol, Boston, MA USA Ikena Oncol, Boston, MA USAEcsedy, Jeffrey论文数: 0 引用数: 0 h-index: 0机构: Ikena Oncol, Boston, MA USA Ikena Oncol, Boston, MA USAMcGovern, Karen论文数: 0 引用数: 0 h-index: 0机构: Ikena Oncol, Boston, MA USA Ikena Oncol, Boston, MA USACastro, Alfredo C.论文数: 0 引用数: 0 h-index: 0机构: Ikena Oncol, Boston, MA USA Ikena Oncol, Boston, MA USA
- [2] The Glutaminase Inhibitor Compound 968 Exhibits Potent In vitro and In vivo Anti-tumor Effects in Endometrial CancerANTI-CANCER AGENTS IN MEDICINAL CHEMISTRY, 2023, 23 (02) : 210 - 221Guo, Hui论文数: 0 引用数: 0 h-index: 0机构: Shandong First Med Univ & Shandong Acad Med Sci, Shandong Canc Hosp & Inst, Dept Gynecol Oncol, Jinan, Shandong, Peoples R China Shandong First Med Univ & Shandong Acad Med Sci, Shandong Canc Hosp & Inst, Dept Gynecol Oncol, Jinan, Shandong, Peoples R ChinaLi, Wanhu论文数: 0 引用数: 0 h-index: 0机构: Shandong First Med Univ & Shandong Acad Med Sci, Shandong Canc Hosp & Inst, Dept Med Imaging, Jinan, Shandong, Peoples R China Shandong First Med Univ & Shandong Acad Med Sci, Shandong Canc Hosp & Inst, Dept Gynecol Oncol, Jinan, Shandong, Peoples R ChinaPan, Guoyou论文数: 0 引用数: 0 h-index: 0机构: Shandong First Med Univ & Shandong Acad Med Sci, Shandong Canc Hosp & Inst, Dept Gynecol Oncol, Jinan, Shandong, Peoples R China Shandong First Med Univ & Shandong Acad Med Sci, Shandong Canc Hosp & Inst, Dept Gynecol Oncol, Jinan, Shandong, Peoples R ChinaWang, Cong论文数: 0 引用数: 0 h-index: 0机构: Shandong First Med Univ & Shandong Acad Med Sci, Shandong Canc Hosp & Inst, Dept Gynecol Oncol, Jinan, Shandong, Peoples R China Shandong First Med Univ & Shandong Acad Med Sci, Shandong Canc Hosp & Inst, Dept Gynecol Oncol, Jinan, Shandong, Peoples R ChinaLi, Dapeng论文数: 0 引用数: 0 h-index: 0机构: Shandong First Med Univ & Shandong Acad Med Sci, Shandong Canc Hosp & Inst, Dept Gynecol Oncol, Jinan, Shandong, Peoples R China Shandong First Med Univ & Shandong Acad Med Sci, Shandong Canc Hosp & Inst, Dept Gynecol Oncol, Jinan, Shandong, Peoples R ChinaLiu, Naifu论文数: 0 引用数: 0 h-index: 0机构: Shandong First Med Univ & Shandong Acad Med Sci, Shandong Canc Hosp & Inst, Dept Gynecol Oncol, Jinan, Shandong, Peoples R China Shandong First Med Univ & Shandong Acad Med Sci, Shandong Canc Hosp & Inst, Dept Gynecol Oncol, Jinan, Shandong, Peoples R ChinaSheng, Xiugui论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Med Sci & Peking Union Med Coll, Canc Hosp, Natl Canc Ctr, Natl Clin Res Ctr Canc, Shenzhen, Peoples R China Chinese Acad Med Sci & Peking Union Med Coll, Shenzhen Hosp, Shenzhen, Peoples R China Shandong First Med Univ & Shandong Acad Med Sci, Shandong Canc Hosp & Inst, Dept Gynecol Oncol, Jinan, Shandong, Peoples R ChinaYuan, Lingqin论文数: 0 引用数: 0 h-index: 0机构: Shandong First Med Univ & Shandong Acad Med Sci, Shandong Canc Hosp & Inst, Dept Gynecol Oncol, Jinan, Shandong, Peoples R China Shandong First Med Univ & Shandong Acad Med Sci, Shandong Canc Hosp & Inst, Dept Gynecol Oncol, Jinan, Shandong, Peoples R China
- [3] Discovery of novel and potent TEAD inhibitors, orally available small molecules with anti-tumor activity in hippo pathway-dysregulated cancersMOLECULAR CANCER THERAPEUTICS, 2023, 22 (12)Moon, Sungho论文数: 0 引用数: 0 h-index: 0Cho, Seon Yeon论文数: 0 引用数: 0 h-index: 0Kim, Minhye论文数: 0 引用数: 0 h-index: 0Beak, Soojeong论文数: 0 引用数: 0 h-index: 0Kim, Jinhyuk论文数: 0 引用数: 0 h-index: 0Kim, Yongchan论文数: 0 引用数: 0 h-index: 0Park, Sungil论文数: 0 引用数: 0 h-index: 0Kim, Jung-In论文数: 0 引用数: 0 h-index: 0Kim, Hanseong论文数: 0 引用数: 0 h-index: 0Lee, In Sang论文数: 0 引用数: 0 h-index: 0No, Kyoung Tai论文数: 0 引用数: 0 h-index: 0
- [4] Discovery and characterization of a new potent orally available CdC7 inhibitor with anti-tumor activityEJC SUPPLEMENTS, 2008, 6 (12): : 116 - 116Montagnoli, A.论文数: 0 引用数: 0 h-index: 0机构: Nerviano Med Sci, Cell Biol, Milan, Italy Nerviano Med Sci, Cell Biol, Milan, ItalyVanotti, E.论文数: 0 引用数: 0 h-index: 0机构: Nerviano Med Sci, Chem, Milan, Italy Nerviano Med Sci, Cell Biol, Milan, ItalyRainoldi, S.论文数: 0 引用数: 0 h-index: 0机构: Nerviano Med Sci, Cell Biol, Milan, Italy Nerviano Med Sci, Cell Biol, Milan, ItalyMarchesi, V.论文数: 0 引用数: 0 h-index: 0机构: Nerviano Med Sci, Cell Biol, Milan, Italy Nerviano Med Sci, Cell Biol, Milan, ItalyCiavolella, A.论文数: 0 引用数: 0 h-index: 0机构: Nerviano Med Sci, Cell Biol, Milan, Italy Nerviano Med Sci, Cell Biol, Milan, ItalyCroci, V.论文数: 0 引用数: 0 h-index: 0机构: Nerviano Med Sci, Pharmacol, Milan, Italy Nerviano Med Sci, Cell Biol, Milan, ItalyPatton, V.论文数: 0 引用数: 0 h-index: 0机构: Nerviano Med Sci, Pharmacol, Milan, Italy Nerviano Med Sci, Cell Biol, Milan, ItalyAlbanese, C.论文数: 0 引用数: 0 h-index: 0机构: Nerviano Med Sci, Cell Biol, Milan, Italy Nerviano Med Sci, Cell Biol, Milan, ItalySantocanale, C.论文数: 0 引用数: 0 h-index: 0机构: Univ Ireland, Galway, Ireland Nerviano Med Sci, Cell Biol, Milan, ItalyMoll, J.论文数: 0 引用数: 0 h-index: 0机构: Nerviano Med Sci, Cell Biol, Milan, Italy Nerviano Med Sci, Cell Biol, Milan, Italy
- [5] In vitro and in vivo anti-tumor activity of ARQ 751, a potent and selective AKT inhibitorCANCER RESEARCH, 2016, 76Yu, Yi论文数: 0 引用数: 0 h-index: 0Savage, Ronald E.论文数: 0 引用数: 0 h-index: 0Eathiraj, Sudharshan论文数: 0 引用数: 0 h-index: 0Hall, Terence论文数: 0 引用数: 0 h-index: 0Schwartz, Brian论文数: 0 引用数: 0 h-index: 0Abbadessa, Giovanni论文数: 0 引用数: 0 h-index: 0
- [6] Liraglutide exhibits potential anti-tumor effects on the progression of intrahepatic cholangiocarcinoma, in vitro and in vivoSCIENTIFIC REPORTS, 2024, 14 (01):Trakoonsenathong, Ronnakrit论文数: 0 引用数: 0 h-index: 0机构: Khon Kaen Univ, Cho Kalaphruek Excellent Res Project Med Students, Fac Med, Khon Kaen, Thailand Khon Kaen Univ, Dept Biochem, Fac Med, Khon Kaen 40002, Thailand Khon Kaen Univ, Cho Kalaphruek Excellent Res Project Med Students, Fac Med, Khon Kaen, ThailandKunprom, Waritta论文数: 0 引用数: 0 h-index: 0机构: Khon Kaen Univ, Dept Pathol, Fac Med, Khon Kaen, Thailand Khon Kaen Univ, Cho Kalaphruek Excellent Res Project Med Students, Fac Med, Khon Kaen, Thailand论文数: 引用数: h-index:机构:Yueangchantuek, Padcharee论文数: 0 引用数: 0 h-index: 0机构: Khon Kaen Univ, Dept Biochem, Fac Med, Khon Kaen 40002, Thailand Khon Kaen Univ, Cho Kalaphruek Excellent Res Project Med Students, Fac Med, Khon Kaen, ThailandPimkeeree, Paslada论文数: 0 引用数: 0 h-index: 0机构: Khon Kaen Univ, Dept Biochem, Fac Med, Khon Kaen 40002, Thailand Naresuan Univ, Fac Med Sci, Phitsanulok, Thailand Khon Kaen Univ, Cho Kalaphruek Excellent Res Project Med Students, Fac Med, Khon Kaen, Thailand论文数: 引用数: h-index:机构:Khawkhiaw, Kullanat论文数: 0 引用数: 0 h-index: 0机构: Khon Kaen Univ, Dept Biochem, Fac Med, Khon Kaen 40002, Thailand Khon Kaen Univ, Cholangiocarcinoma Res Inst, Khon Kaen, Thailand Khon Kaen Univ, Cho Kalaphruek Excellent Res Project Med Students, Fac Med, Khon Kaen, ThailandChiu, Ching-Feng论文数: 0 引用数: 0 h-index: 0机构: Taipei Med Univ, Grad Inst Metab & Obes Sci, Taipei, Taiwan Khon Kaen Univ, Cho Kalaphruek Excellent Res Project Med Students, Fac Med, Khon Kaen, Thailand论文数: 引用数: h-index:机构:论文数: 引用数: h-index:机构:Saengboonmee, Charupong论文数: 0 引用数: 0 h-index: 0机构: Khon Kaen Univ, Cho Kalaphruek Excellent Res Project Med Students, Fac Med, Khon Kaen, Thailand Khon Kaen Univ, Dept Biochem, Fac Med, Khon Kaen 40002, Thailand Khon Kaen Univ, Cholangiocarcinoma Res Inst, Khon Kaen, Thailand Khon Kaen Univ, Cho Kalaphruek Excellent Res Project Med Students, Fac Med, Khon Kaen, Thailand
- [7] Novel small molecule inhibitors of p97 demonstrate anti-tumor effects in vitro and in vivoMOLECULAR BIOLOGY OF THE CELL, 2013, 24Anderson, D.论文数: 0 引用数: 0 h-index: 0机构: Cleave Biosci, Burlingame, CA USA Cleave Biosci, Burlingame, CA USADjakovic, S.论文数: 0 引用数: 0 h-index: 0机构: Cleave Biosci, Burlingame, CA USA Cleave Biosci, Burlingame, CA USAKissvonsoly, S.论文数: 0 引用数: 0 h-index: 0机构: Cleave Biosci, Burlingame, CA USA Cleave Biosci, Burlingame, CA USALe Moigne, R.论文数: 0 引用数: 0 h-index: 0机构: Cleave Biosci, Burlingame, CA USA Cleave Biosci, Burlingame, CA USARice, J.论文数: 0 引用数: 0 h-index: 0机构: Cleave Biosci, Burlingame, CA USA Cleave Biosci, Burlingame, CA USARolfe, M.论文数: 0 引用数: 0 h-index: 0机构: Cleave Biosci, Burlingame, CA USA Cleave Biosci, Burlingame, CA USASoriano, F.论文数: 0 引用数: 0 h-index: 0机构: Cleave Biosci, Burlingame, CA USA Cleave Biosci, Burlingame, CA USAValle, E.论文数: 0 引用数: 0 h-index: 0机构: Cleave Biosci, Burlingame, CA USA Cleave Biosci, Burlingame, CA USAWang, J.论文数: 0 引用数: 0 h-index: 0机构: Cleave Biosci, Burlingame, CA USA Cleave Biosci, Burlingame, CA USAWong, S.论文数: 0 引用数: 0 h-index: 0机构: Cleave Biosci, Burlingame, CA USA Cleave Biosci, Burlingame, CA USAWustrow, D.论文数: 0 引用数: 0 h-index: 0机构: Cleave Biosci, Burlingame, CA USA Cleave Biosci, Burlingame, CA USAYakes, M.论文数: 0 引用数: 0 h-index: 0机构: Cleave Biosci, Burlingame, CA USA Cleave Biosci, Burlingame, CA USAYao, B.论文数: 0 引用数: 0 h-index: 0机构: Cleave Biosci, Burlingame, CA USA Cleave Biosci, Burlingame, CA USAZhou, H-J.论文数: 0 引用数: 0 h-index: 0机构: Cleave Biosci, Burlingame, CA USA Cleave Biosci, Burlingame, CA USA
- [8] AP24534: an orally active kinase inhibitor that targets multiple pro-angiogenic receptors and exhibits potent anti-tumor activity in vivoEJC SUPPLEMENTS, 2008, 6 (12): : 174 - 174Rivera, V. M.论文数: 0 引用数: 0 h-index: 0DiRenzo, R.论文数: 0 引用数: 0 h-index: 0Berk, L.论文数: 0 引用数: 0 h-index: 0Wardwell, S.论文数: 0 引用数: 0 h-index: 0Ning, Y.论文数: 0 引用数: 0 h-index: 0Narasimhan, N. I.论文数: 0 引用数: 0 h-index: 0Xu, Q.论文数: 0 引用数: 0 h-index: 0Shakespeare, W. C.论文数: 0 引用数: 0 h-index: 0Wang, F.论文数: 0 引用数: 0 h-index: 0Clackson, T.论文数: 0 引用数: 0 h-index: 0
- [9] L-4, a Well-Tolerated and Orally Active Inhibitor of Hedgehog Pathway, Exhibited Potent Anti-tumor Effects Against Medulloblastoma in vitro and in vivoFRONTIERS IN PHARMACOLOGY, 2019, 10Zhu, Mingfei论文数: 0 引用数: 0 h-index: 0机构: East China Normal Univ, Shanghai Engn Res Ctr Mol Therapeut & New Drug De, Sch Chem & Mol Engn, Shanghai, Peoples R China East China Normal Univ, Shanghai Engn Res Ctr Mol Therapeut & New Drug De, Sch Chem & Mol Engn, Shanghai, Peoples R ChinaWang, Hong论文数: 0 引用数: 0 h-index: 0机构: East China Normal Univ, Shanghai Engn Res Ctr Mol Therapeut & New Drug De, Sch Chem & Mol Engn, Shanghai, Peoples R China East China Normal Univ, Shanghai Engn Res Ctr Mol Therapeut & New Drug De, Sch Chem & Mol Engn, Shanghai, Peoples R ChinaWang, Chenglin论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Sch Pharm, Dept Med Chem, Shanghai, Peoples R China East China Normal Univ, Shanghai Engn Res Ctr Mol Therapeut & New Drug De, Sch Chem & Mol Engn, Shanghai, Peoples R ChinaFang, Yanfen论文数: 0 引用数: 0 h-index: 0机构: East China Normal Univ, Shanghai Engn Res Ctr Mol Therapeut & New Drug De, Sch Chem & Mol Engn, Shanghai, Peoples R China East China Normal Univ, Shanghai Engn Res Ctr Mol Therapeut & New Drug De, Sch Chem & Mol Engn, Shanghai, Peoples R ChinaZhu, Tong论文数: 0 引用数: 0 h-index: 0机构: East China Normal Univ, Shanghai Engn Res Ctr Mol Therapeut & New Drug De, Sch Chem & Mol Engn, Shanghai, Peoples R China East China Normal Univ, Shanghai Engn Res Ctr Mol Therapeut & New Drug De, Sch Chem & Mol Engn, Shanghai, Peoples R ChinaZhao, Weili论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Sch Pharm, Dept Med Chem, Shanghai, Peoples R China East China Normal Univ, Shanghai Engn Res Ctr Mol Therapeut & New Drug De, Sch Chem & Mol Engn, Shanghai, Peoples R ChinaDong, Xiaochun论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Sch Pharm, Dept Med Chem, Shanghai, Peoples R China East China Normal Univ, Shanghai Engn Res Ctr Mol Therapeut & New Drug De, Sch Chem & Mol Engn, Shanghai, Peoples R ChinaZhang, Xiongwen论文数: 0 引用数: 0 h-index: 0机构: East China Normal Univ, Shanghai Engn Res Ctr Mol Therapeut & New Drug De, Sch Chem & Mol Engn, Shanghai, Peoples R China East China Normal Univ, Shanghai Engn Res Ctr Mol Therapeut & New Drug De, Sch Chem & Mol Engn, Shanghai, Peoples R China
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