Convenient synthesis of (4R,5R)-4,5-bis(aminomethyl)-2-isopropyl-1,3-dioxolane

被引：0
|
作者：
Jian Jiang
机构：
来源：
Chinese Chemical Letters | 2007年 / 07期
关键词：
Heptaplatin; Aminomethyl; Intermediate; Anticancer drug;
D O I：
暂无
中图分类号：
O621.3 [有机合成化学];
学科分类号：
070303 ; 081704 ;
摘要：
A convenient approach for the preparation of (4R,5R)-4,5-bis(aminomethyl)-2-isopropyl-1,3-dioxolane is described. The target compound via two steps is synthesized from diethyl-2,3-O-isobutylidene-D-tartrate, through ammonolysis and reduction.
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页码：783 / 784
页数：2
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