Copper-catalyzed N-arylation of 2-arylindoles with aryl halides

被引：1

作者：

Wei Liu ^{[1
]}

Li-Ya Han ^{[1
]}

Rui-Li Liu ^{[1
]}

Li-Ge Xu ^{[1
]}

Yan-Lan Bi ^{[1
]}

机构：

[1] College of Food Science and Technology,Henan University of Technology

来源：

Chinese Chemical Letters | 2014年 / 25卷 / 09期

基金：

中国国家自然科学基金;

关键词：

2-Arylindoles; Aryl halides; N-Arylation; Copper;

D O I：

暂无

中图分类号：

O621.251 [];

学科分类号：

070303 ; 081704 ;

摘要：

10 mol% CuI combined with the DMEDA ligand can efficiently catalyze the N-arylation of 2-arylindoles with aryl iodides and aryl bromides in good to excellent yields.The aryl halides bearing electron-rich or electron-deficient functional groups can be well tolerated under this mild reaction conditions.

引用

页码：1240 / 1243

页数：4

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