An Effective N-Ligand for Copper-Catalyzed N-Arylation of Triazole

被引:0
|
作者
Yang, Yan [1 ]
Jin, Yong-Sheng [1 ]
Hu, Hong-Gang [1 ]
Zhao, Qing-Jie [1 ]
Zou, Yan [1 ]
Wu, Qui-Ye [1 ]
机构
[1] Second Mil Med Univ, Dept Organ Chem, Sch Pharm, Shanghai 200433, Peoples R China
基金
中国国家自然科学基金;
关键词
N-Ligand; C-N Bond cross-coupling; Copper-catalyzed; 1H-1,2,4-Triazole; AMINATION;
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
An effective N-ligand for copper-catalyzed N-arylation of 1H-1,2,4-triazole has been developed. In the presence of Cu2O, Cs2CO3, N-ligand-B. 1H-1,2,4-triazole were coupled with toluence to afford the corresponding products in moderate condition and with excellent yields.
引用
收藏
页码:7435 / 7437
页数:3
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