Discovery of KRas G12C-IN-3 and Pomalidomide-based PROTACs as degraders of endogenous KRAS G12C with potent anticancer activity (vol 117, 105447, 2021)

被引:0
|
作者
Li, Ling [1 ]
Wu, Yinrong [1 ]
Yang, Zichao [1 ]
Xu, Chenglong [1 ]
Zhao, Huiting [1 ]
Liu, Jin [1 ]
Chen, Jingxuan [1 ]
Chen, Jianjun [1 ]
机构
[1] Southern Med Univ, Sch Pharmaceut Sci, Guangdong Prov Key Lab New Drug Screening, Guangzhou 510515, Peoples R China
关键词
D O I
10.1016/j.bioorg.2024.107616
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
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页数:2
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