SYNTHESIS OF A NOVEL TETRACYCLIC HETEROCYCLE - 1-CARBOXY-13-OXO-[1,2,3]TRIAZOLO[1',5'/4,3][1,4]DIAZEPINO[6,7-C]CHROMANE, USING SALICYLALDEHYDE AS A STARTING MATERIAL

被引：12

作者：

KELLABENNANI, AE

SOUFIAOUI, M

KERBAL, A

FKIHTETOUANI, S

BITIT, N

机构：

[1] FAC SCI RABAT,CHIM PLANTES & SYNTH ORGAN & BIOORGAN LAB,RABAT,MOROCCO

[2] FAC SCI DHAR MAHRAZ,CHIM ORGAN LAB,ATLAS FES,MOROCCO

来源：

TETRAHEDRON | 1995年 / 51卷 / 40期

关键词：

D O I：

10.1016/0040-4020(95)00668-X

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A nine-step synthesis of the potentially biologically active tide compound, 9,has been achieved starting from salicylaldehyde and involving two 1,3-dipolar cycloaddition reactions and a lactamisation reaction. The cis configuration of compound 9 resulted from that of compound 4 which was confirmed by X-ray crystallography.

引用

页码：10923 / 10928

页数：6

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