CHEMICAL MODIFICATION OF RAT CEREBRAL-CORTEX M1 MUSCARINIC RECEPTORS - ROLE OF HISTIDYL RESIDUES IN ANTAGONIST AND AGONIST BINDING

被引:4
|
作者
VANKOPPEN, CJ
SOKOLOVSKY, M
机构
关键词
D O I
10.1016/S0006-291X(88)80474-1
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:1069 / 1073
页数:5
相关论文
共 50 条
  • [41] PURIFICATION AND PROPERTIES OF M1-TOXIN, A SPECIFIC ANTAGONIST OF M1 MUSCARINIC RECEPTORS
    MAX, SI
    LIANG, JS
    POTTER, LT
    JOURNAL OF NEUROSCIENCE, 1993, 13 (10): : 4293 - 4300
  • [42] STABLE ALLOSTERIC BINDING OF M1-TOXIN TO M1 MUSCARINIC RECEPTORS
    MAX, SI
    LIANG, JS
    POTTER, LT
    MOLECULAR PHARMACOLOGY, 1993, 44 (06) : 1171 - 1175
  • [43] MUSCARINIC M1 RECEPTORS ARE PHOSPHORYLATED IN CHO CELLS FOLLOWING AGONIST STIMULATION
    WAUGH, MG
    BURFORD, NT
    NAHORSKI, SR
    TOBIN, AB
    BRITISH JOURNAL OF PHARMACOLOGY, 1995, 114 : P143 - P143
  • [44] EFFECTS OF THE CA-2+-ANTAGONISTS NIFEDIPINE, VERAPAMIL, FLUNARIZINE AND OF THE CALMODULIN ANTAGONIST TRIFLUOPERAZINE ON MUSCARINIC CHOLINERGIC RECEPTORS IN RAT CEREBRAL-CORTEX
    POPOVA, J
    STANEVASTOYTCHEVA, D
    MUTAFOVA, V
    GENERAL PHARMACOLOGY, 1990, 21 (03): : 317 - 319
  • [45] Spatio-temporal distribution of M1/M2 muscarinic cholinergic receptors in rat cerebral cortex after focal photothrombotic stroke
    Rogozinska, K.
    Aleksy, M.
    Skangiel-Kramska, J.
    JOURNAL OF NEUROCHEMISTRY, 2007, 101 : 44 - 44
  • [46] EFFECTS OF DEPOLARIZING AGENTS AND NA+-CHANNEL INHIBITORS ON LIGAND-BINDING TO MUSCARINIC RECEPTORS FROM RAT CEREBRAL-CORTEX
    HEDLUND, B
    ACTA CHEMICA SCANDINAVICA SERIES B-ORGANIC CHEMISTRY AND BIOCHEMISTRY, 1987, 41 (09): : 686 - 693
  • [47] Immunolocalization of muscarinic M1 receptor in the rat medial prefrontal cortex
    Oda, Satoko
    Tsuneoka, Yousuke
    Yoshida, Sachine
    Adachi-Akahane, Satomi
    Ito, Masanori
    Kuroda, Masaru
    Funato, Hiromasa
    JOURNAL OF COMPARATIVE NEUROLOGY, 2018, 526 (08) : 1329 - 1350
  • [48] CLOZAPINE IS A POTENT AGONIST AT HUMAN M4 MUSCARINIC RECEPTORS AND AN ANTAGONIST AT M1, M2, M3, AND M5 RECEPTORS
    LISTON, D
    WARD, KM
    JONES, SB
    ZORN, SH
    LIFE SCIENCES, 1995, 56 (11-12) : 1018 - 1018
  • [49] A SELECTIVE ROLE OF MUSCARINIC RECEPTORS IN K+-EVOKED INOSITOL TETRAKISPHOSPHATE ACCUMULATION IN CEREBRAL-CORTEX
    BAIRD, JG
    NAHORSKI, SR
    BRITISH JOURNAL OF PHARMACOLOGY, 1988, 94 : P395 - P395
  • [50] EFFECTS OF THE METHYLXANTHINE DERIVATIVE PENTOXIFYLLINE ON BENZODIAZEPINE AND MUSCARINIC BINDING-SITES IN RAT CEREBRAL-CORTEX
    LOWENSTEIN, PR
    AGUILAR, JSO
    SABATO, UC
    ACTA PHYSIOLOGICA ET PHARMACOLOGICA LATINOAMERICANA, 1985, 35 (04): : 431 - 439