CHEMICAL MODIFICATION OF RAT CEREBRAL-CORTEX M1 MUSCARINIC RECEPTORS - ROLE OF HISTIDYL RESIDUES IN ANTAGONIST AND AGONIST BINDING

被引:4
|
作者
VANKOPPEN, CJ
SOKOLOVSKY, M
机构
关键词
D O I
10.1016/S0006-291X(88)80474-1
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:1069 / 1073
页数:5
相关论文
共 50 条
  • [21] THE EFFECT OF PARA-CHLOROMERCURIBENZOATE ON STRUCTURE-BINDING RELATIONSHIPS OF MUSCARINIC RECEPTORS IN THE RAT CEREBRAL-CORTEX
    BIRDSALL, NJM
    BURGEN, ASV
    HULME, EC
    WONG, EHF
    BRITISH JOURNAL OF PHARMACOLOGY, 1983, 80 (01) : 197 - 204
  • [22] Muscarinic M1 and M3 receptors in rat striatum:: A binding study
    De la Vega, MT
    Nunez, A
    Arias-Montano, JA
    ARCHIVES OF MEDICAL RESEARCH, 1997, 28 (04): : 493 - 497
  • [23] DETERMINATION OF MUSCARINIC AGONIST POTENCIES AT M1 AND M2 MUSCARINIC RECEPTORS IN A MODIFIED PITHED RAT PREPARATION
    ANGELI, P
    BRASILI, L
    CANTALAMESSA, F
    MARUCCI, G
    WESS, J
    NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1990, 342 (06) : 625 - 629
  • [24] Mutant M1 muscarinic receptors with enhanced agonist activity
    Huang, XP
    Williams, FE
    Peseckis, SM
    Messer, WS
    LIFE SCIENCES, 1999, 64 (6-7) : 563 - 563
  • [25] AGONIST-INDUCED PHOSPHORYLATION OF M1 MUSCARINIC RECEPTORS
    WAUGH, MG
    NAHORSKI, SR
    TOBIN, AB
    LIFE SCIENCES, 1995, 56 (11-12) : 1026 - 1026
  • [26] TEMPERATURE EFFECT ON SUBCLASSES OF MUSCARINIC RECEPTORS IN RAT COLON, HEART AND CEREBRAL-CORTEX
    MUZIO, F
    MALANDRINO, S
    FERRARI, M
    TONON, G
    LIFE SCIENCES, 1986, 39 (04) : 365 - 371
  • [27] EFFECT OF ELECTROCONVULSIVE SHOCK ON MUSCARINIC CHOLINERGIC RECEPTORS IN RAT CEREBRAL-CORTEX AND HIPPOCAMPUS
    LERER, B
    STANLEY, M
    DEMETRIOU, S
    GERSHON, S
    JOURNAL OF NEUROCHEMISTRY, 1983, 41 (06) : 1680 - 1683
  • [28] AGONIST AND ANTAGONIST BINDING TO RAT-BRAIN MUSCARINIC RECEPTORS - INFLUENCE OF AGING
    GURWITZ, D
    EGOZI, Y
    HENIS, YI
    KLOOG, Y
    SOKOLOVSKY, M
    NEUROBIOLOGY OF AGING, 1987, 8 (02) : 115 - 122
  • [29] THE BINDING OF A 2-CHLOROETHYLAMINE DERIVATIVE OF OXOTREMORINE (BM-123) TO MUSCARINIC RECEPTORS IN THE RAT CEREBRAL-CORTEX
    EHLERT, FJ
    JENDEN, DJ
    MOLECULAR PHARMACOLOGY, 1985, 28 (02) : 107 - 119
  • [30] HEXAHYDRODIFENIDOL DOES NOT DISTINGUISH AMONG M1 RECEPTORS IN RAT CEREBRAL-CORTEX, HIPPOCAMPUS AND SUPERIOR CERVICAL-GANGLION
    FREEDMAN, SB
    FIELD, JL
    GILBERT, MJ
    NEWBERRY, NR
    EUROPEAN JOURNAL OF PHARMACOLOGY, 1989, 167 (03) : 411 - 414