INVIVO AND INVITRO PHARMACOLOGY OF SR48,968 AS TACHYKININ NK-2 RECEPTOR ANTAGONIST

被引:0
|
作者
GIULIANI, S [1 ]
PATACCHINI, R [1 ]
GIACHETTI, A [1 ]
MAGGI, CA [1 ]
机构
[1] A MENARINI PHARMACEUT,DEPT PHARMACOL,I-50131 FLORENCE,ITALY
关键词
D O I
暂无
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
引用
收藏
页码:S63 / S63
页数:1
相关论文
共 50 条
  • [31] PHARMACOLOGY OF CP-99,994 - A NONPEPTIDE ANTAGONIST OF THE TACHYKININ NK1 RECEPTOR
    MCLEAN, S
    GANONG, A
    SEYMOUR, PA
    SNIDER, RM
    DESAI, MC
    ROSEN, T
    BRYCE, DK
    LONGO, KP
    REYNOLDS, LS
    ROBINSON, G
    SCHMIDT, AW
    SIOK, C
    HEYM, J
    REGULATORY PEPTIDES, 1992, : S120 - S120
  • [32] Monocyclic human tachykinin NK-2 receptor antagonists as evolution of a potent bicyclic antagonist: QSAR and site-directed mutagenesis studies
    Giolitti, A
    Altamura, M
    Bellucci, F
    Giannotti, D
    Meini, S
    Patacchini, R
    Rotondaro, L
    Zappitelli, S
    Maggi, CA
    JOURNAL OF MEDICINAL CHEMISTRY, 2002, 45 (16) : 3418 - 3429
  • [33] ACTIVITY OF SPANTIDE-I AND SPANTIDE-II AT VARIOUS TACHYKININ RECEPTORS AND NK-2 TACHYKININ RECEPTOR SUBTYPES
    MAGGI, CA
    PATACCHINI, R
    FENG, DM
    FOLKERS, K
    EUROPEAN JOURNAL OF PHARMACOLOGY, 1991, 199 (01) : 127 - 129
  • [34] A versatile synthesis of a beta-turn peptidomimetic scaffold: An approach towards a designed model antagonist of the tachykinin NK-2 receptor.
    Hanessian, S
    McNaughtonSmith, G
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1996, 6 (13) : 1567 - 1572
  • [35] N-TERMINAL TRUNCATED ANALOGS OF MEN 10376 AS TACHYKININ NK-2 RECEPTOR ANTAGONISTS
    QUARTARA, L
    PATACCHINI, R
    GIULIANI, S
    RENZETTI, AR
    ROVERO, P
    MAGGI, CA
    LIFE SCIENCES, 1992, 51 (25) : 1929 - 1936
  • [36] Antigen inhalation unmasks NK-2 tachykinin receptor-mediated responses in vagal afferents
    Moore, KA
    Undem, BJ
    Weinreich, D
    AMERICAN JOURNAL OF RESPIRATORY AND CRITICAL CARE MEDICINE, 2000, 161 (01) : 232 - 236
  • [37] SR-142801, THE FIRST POTENT NONPEPTIDE ANTAGONIST OF THE TACHYKININ NK3 RECEPTOR
    EMONDSALT, X
    BICHON, D
    DUCOUX, JP
    HEAULME, M
    MILOUX, B
    PONCELET, M
    PROIETTO, V
    VANBROECK, D
    VILAIN, P
    NELIAT, G
    SOUBRIE, P
    LEFUR, G
    BRELIERE, JC
    LIFE SCIENCES, 1994, 56 (01) : PL27 - PL32
  • [38] CONFORMATIONALLY CONSTRAINED TACHYKININ ANALOGS - POTENT AND HIGHLY SELECTIVE NEUROKININ NK-2 RECEPTOR AGONISTS
    DEAL, MJ
    HAGAN, RM
    IRELAND, SJ
    JORDAN, CC
    MCELROY, AB
    PORTER, B
    ROSS, BC
    STEPHENSSMITH, M
    WARD, P
    JOURNAL OF MEDICINAL CHEMISTRY, 1992, 35 (22) : 4195 - 4204
  • [39] PHARMACOLOGY OF GR203040, A POTENT AND SELECTIVE NONPEPTIDE TACHYKININ NK1 RECEPTOR ANTAGONIST
    BEATTIE, DT
    CONNER, HE
    HAWCOCK, AB
    PERREN, MJ
    WARD, P
    BRITISH JOURNAL OF PHARMACOLOGY, 1995, 116 : P37 - P37
  • [40] The peripheral NK-1/NK-2 receptor antagonist MDL 105,172A inhibits tachykinin-mediated respiratory effects in guinea-pigs
    Kudlacz, EM
    Knippenberg, RW
    Shatzer, SA
    Kehne, JH
    McCloskey, TC
    Burkholder, TP
    JOURNAL OF AUTONOMIC PHARMACOLOGY, 1997, 17 (02): : 109 - 119