INHIBITION OF GLYCINE AND GABA RECEPTOR-BINDING BY SEVERAL OPIATE AGONISTS AND ANTAGONISTS

被引:31
|
作者
GOLDINGER, A [1 ]
MULLER, WE [1 ]
WOLLERT, U [1 ]
机构
[1] UNIV MAINZ,INST PHARMAKOL,D-6500 MAINZ,FED REP GER
来源
GENERAL PHARMACOLOGY | 1981年 / 12卷 / 06期
关键词
D O I
10.1016/0306-3623(81)90073-2
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
下载
收藏
页码:477 / 479
页数:3
相关论文
共 50 条
  • [41] Positive Modulation of the Glycine Receptor by Means of Glycine Receptor-Binding Aptamers
    Shalaly, Nancy Dekki
    Aneiros, Eduardo
    Blank, Michael
    Mueller, Johan
    Nyman, Eva
    Blind, Michael
    Dabrowski, Michael A.
    Andersson, Christin V.
    Sandberg, Kristian
    JOURNAL OF BIOMOLECULAR SCREENING, 2015, 20 (09) : 1112 - 1123
  • [42] GABA(A) RECEPTOR AGONISTS, PARTIAL AGONISTS, AND ANTAGONISTS - DESIGN AND THERAPEUTIC PROSPECTS
    KROGSGAARDLARSEN, P
    FROLUND, B
    JORGENSEN, FS
    SCHOUSBOE, A
    JOURNAL OF MEDICINAL CHEMISTRY, 1994, 37 (16) : 2489 - 2505
  • [43] DIFFERENTIAL EFFECT OF HUMORAL ENDORPHIN ON THE BINDING OF OPIATE AGONISTS AND ANTAGONISTS
    SARNE, Y
    ITZHAK, Y
    KEREN, O
    EUROPEAN JOURNAL OF PHARMACOLOGY, 1982, 81 (02) : 227 - 235
  • [44] INTERACTIONS OF AGONISTS AND ANTAGONISTS WITH A NOVEL TYPE OF GABA RECEPTOR
    MITCHELL, R
    BIOCHEMICAL PHARMACOLOGY, 1982, 31 (16) : 2684 - 2686
  • [45] PRETREATMENT WITH GABA AND MODULATORY LIGANDS ENHANCES GABA RECEPTOR-BINDING
    MAKSAY, G
    TICKU, MK
    EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 104 (1-2) : 185 - 188
  • [46] REVERSAL BY BOVINE SERUM-ALBUMIN OF PHOSPHOLIPASE-A INHIBITION OF OPIATE RECEPTOR-BINDING
    LIN, HK
    SIMON, EJ
    FEDERATION PROCEEDINGS, 1978, 37 (03) : 238 - 238
  • [47] METHADONE BINDING AT NON-OPIATE RECEPTOR-BINDING SITES
    CIOFALO, FR
    RESEARCH COMMUNICATIONS IN CHEMICAL PATHOLOGY AND PHARMACOLOGY, 1979, 24 (03): : 419 - 430
  • [48] GABA(A) and GABA(B) receptor agonists, partial agonists, antagonists and modulators: design and therapeutic prospects
    KrogsgaardLarsen, P
    Frolund, B
    Kristiansen, U
    Frydenvang, K
    Ebert, B
    EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 1997, 5 (06) : 355 - 384
  • [49] OPIATE RECEPTOR CHANGES AFTER CHRONIC EXPOSURE TO AGONISTS AND ANTAGONISTS
    ZADINA, JE
    KASTIN, AJ
    HARRISON, LM
    GE, LJ
    CHANG, SL
    DIVERSITY OF INTERACTING RECEPTORS, 1995, 757 : 353 - 361
  • [50] COMPARISON OF RECEPTOR-BINDING CHARACTERISTICS OF OPIATE AGONISTS INTERACTING WITH MU-RECEPTORS OR KAPPA-RECEPTORS
    KOSTERLITZ, HW
    LESLIE, FM
    BRITISH JOURNAL OF PHARMACOLOGY, 1978, 64 (04) : 607 - 614