RETINOBENZOIC ACIDS .4. CONFORMATION OF AROMATIC AMIDES WITH RETINOIDAL ACTIVITY - IMPORTANCE OF TRANS-AMIDE STRUCTURE FOR THE ACTIVITY

被引：84

作者：

KAGECHIKA, H ^{[1
]}

HIMI, T ^{[1
]}

KAWACHI, E ^{[1
]}

SHUDO, K ^{[1
]}

机构：

[1] UNIV TOKYO,FAC PHARMACEUT SCI,7-3-1 HONGO,BUNKYO KU,TOKYO 113,JAPAN

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1989年 / 32卷 / 10期

关键词：

D O I：

10.1021/jm00130a011

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：2292 / 2296

页数：5

共 34 条

[31] STUDIES ON BETA-LACTAM ANTIBIOTICS .4. STRUCTURE-ACTIVITY-RELATIONSHIPS OF 7-BETA-[(Z)-2-ALKOXYIMINO-2-(2-AMINO-4-THIAZOLYL)ACETAMIDO]-3-CEPHEM-4-CARBOXYLIC ACIDS
TAKAYA, T
TAKASUGI, H
MASUGI, T
KOCHI, H
NAKANO, H
JOURNAL OF ANTIBIOTICS, 1981, 34 (10): : 1357 - 1359
[32] FLUORONAPHTHYRIDINES AS ANTIBACTERIAL AGENTS .4. SYNTHESIS AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF 5-SUBSTITUTED-6-FLUORO-7-(CYCLOALKYLAMINO)-1,4-DIHYDRO-4-OXO-1,8-NAPHTHYRIDINE-3-CARBOXYLIC ACIDS
BOUZARD, D
DICESARE, P
ESSIZ, M
JACQUET, JP
LEDOUSSAL, B
REMUZON, P
KESSLER, RE
FUNGTOMC, J
JOURNAL OF MEDICINAL CHEMISTRY, 1992, 35 (03) : 518 - 525
[33] Studies on quinolone antibacterials .4. Structure-activity relationships of antibacterial activity and side effects for 5- or 8-substituted and 5,8-disubstituted-7-(3-amino-1-pyrrolidinyl)-1-cyclopropyl-1,4-dihydro-4-oxoquinoline-3-carboxylic acids
Yoshida, T
Yamamoto, Y
Orita, H
Kakiuchi, M
Takahashi, Y
Itakura, M
Kado, N
Mitani, K
Yasuda, S
Kato, H
Itoh, Y
CHEMICAL & PHARMACEUTICAL BULLETIN, 1996, 44 (05) : 1074 - 1085
[34] Synthesis and structure-activity relationships of a new model of arylpiperazines.: 4.: 1-[ω-(4-arylpiperazin-1-yl)alkyl]-3-(diphenylmethylene)-2,5-pyrrolidinediones and -3-(9H-fluoren-9-ylidene)-2,5-pyrrolidinediones:: Study of the steric requirements of the terminal amide fragment on 5-HT1A affinity/selectivity
López-Rodríguez, ML
Morcillo, MJ
Rovat, TK
Fernández, E
Vicente, B
Sanz, AM
Hernández, M
Orensanz, L
JOURNAL OF MEDICINAL CHEMISTRY, 1999, 42 (01) : 36 - 49

← 1 2 3 4 →