ANTAGONISTS OF NK2 TACHYKININ RECEPTORS AS A POTENTIAL NEW CLASS OF ANTIBRONCHOSPASTIC AGENTS

被引:6
|
作者
MANZINI, S
机构
[1] Menarini Ricerche Sud, Pharmacology Department, 00040 Pomezia, Roma
来源
GENERAL PHARMACOLOGY | 1994年 / 25卷 / 01期
关键词
D O I
10.1016/0306-3623(94)90002-7
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
[No abstract available]
引用
收藏
页码:1 / 6
页数:6
相关论文
共 50 条
  • [41] Role of tachykinin NK1, NK2 and NK3 receptors in the modulation of visceral hypersensitivity in the rat
    Gaudreau, GA
    Plourde, V
    NEUROSCIENCE LETTERS, 2003, 351 (02) : 59 - 62
  • [42] An investigation of tachykinin NK2 receptor subtypes in the rat
    Matuszek, MA
    Zeng, XP
    Strigas, J
    Burcher, E
    EUROPEAN JOURNAL OF PHARMACOLOGY, 1998, 352 (01) : 103 - 109
  • [43] INVOLVEMENT OF TACHYKININ RECEPTORS (NK1 AND NK2) IN SODIUM METABISULFITE-INDUCED AIRWAY EFFECTS
    SAKAMOTO, T
    TSUKAGOSHI, H
    BARNES, PJ
    CHUNG, KF
    AMERICAN JOURNAL OF RESPIRATORY AND CRITICAL CARE MEDICINE, 1994, 149 (02) : 387 - 391
  • [44] Molecular determinants of neuropeptide-mediated activation mechanisms in tachykinin NK1 and NK2 receptors
    Petersen, Jacob E.
    Pavlovskyi, Artem
    Madsen, Jesper J.
    Schwartz, Thue W.
    Frimurer, Thomas M.
    Olsen, Ole H.
    JOURNAL OF BIOLOGICAL CHEMISTRY, 2024, 300 (12)
  • [45] Design, synthesis, and SAR of tachykinin antagonists:: Modulation of balance in NK1/NK2 receptor antagonist activity
    Albert, JS
    Aharony, D
    Andisik, D
    Barthlow, H
    Bernstein, PR
    Bialecki, RA
    Dedinas, R
    Dembofsky, BT
    Hill, D
    Kirkland, K
    Koether, GM
    Kosmider, BJ
    Ohnmacht, C
    Palmer, W
    Potts, W
    Rumsey, W
    Shen, LH
    Shenvi, A
    Sherwood, S
    Warwick, PJ
    Russell, K
    JOURNAL OF MEDICINAL CHEMISTRY, 2002, 45 (18) : 3972 - 3983
  • [46] AFFINITY OF THE NK2 ANTAGONIST SR 48968 AT NK3-TACHYKININ AND MU-OPIOID RECEPTORS
    BOYLE, SJ
    MANLEY, S
    TANG, KW
    MEECHAM, K
    GUARD, S
    WATLING, KJ
    WOODRUFF, GN
    MCKNIGHT, AT
    BRITISH JOURNAL OF PHARMACOLOGY, 1993, 108 : P24 - P24
  • [47] Role of tachykinin NK1 and NK2 receptors on colonic motility in anesthetized rats: effect of agonists
    Lecci, A
    Tramontana, M
    Giuliani, S
    Maggi, CA
    CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY, 1997, 75 (06) : 582 - 586
  • [48] THE NONPEPTIDE TACHYKININ NK2 RECEPTOR ANTAGONIST SR-48968 INTERACTS WITH HUMAN, BUT NOT RAT, CLONED TACHYKININ NK3 RECEPTORS
    CHUNG, FZ
    WU, LH
    VARTANIAN, MA
    WATLING, KJ
    GUARD, S
    WOODRUFF, GN
    OXENDER, DL
    BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1994, 198 (03) : 967 - 972
  • [49] EVIDENCE FOR HETEROGENEITY OF NK-2 TACHYKININ RECEPTORS BY USING COMPETITIVE ANTAGONISTS
    SANTICIOLI, P
    MAGGI, CA
    PATACCHINI, R
    GIULIANI, S
    ROVERO, P
    REGOLI, D
    MELI, A
    GIACHETTI, A
    EUROPEAN JOURNAL OF PHARMACOLOGY, 1990, 183 (06) : 2141 - 2142
  • [50] Distribution pattern of tachykinin NK2 receptors in human colon:: Involvement in the regulation of intestinal motility
    Jaafari, Nadia
    Khomitch-Baud, Alexandra
    Christen, Marie-Odile
    Jule, Yvon
    JOURNAL OF COMPARATIVE NEUROLOGY, 2007, 503 (03) : 381 - 391