ANTAGONISTS OF NK2 TACHYKININ RECEPTORS AS A POTENTIAL NEW CLASS OF ANTIBRONCHOSPASTIC AGENTS

被引:6
|
作者
MANZINI, S
机构
[1] Menarini Ricerche Sud, Pharmacology Department, 00040 Pomezia, Roma
来源
GENERAL PHARMACOLOGY | 1994年 / 25卷 / 01期
关键词
D O I
10.1016/0306-3623(94)90002-7
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
[No abstract available]
引用
收藏
页码:1 / 6
页数:6
相关论文
共 50 条
  • [1] NK2 ANTAGONISTS AND THE ROLE OF NK2 RECEPTORS
    HAGAN, RM
    BERESFORD, IJM
    ELLIOTT, PJ
    BALL, DI
    SHELDRICK, RLG
    IRELAND, SJ
    PRITCHARD, JM
    MCELROY, AB
    WARD, P
    REGULATORY PEPTIDES, 1992, : S8 - S8
  • [3] Small molecule antagonists of the tachykinin NK2 receptor
    Fattori, D
    Altamura, M
    Maggi, CA
    MINI-REVIEWS IN MEDICINAL CHEMISTRY, 2004, 4 (03) : 331 - 340
  • [4] Glycosyl derivatives of NK2 tachykinin receptor antagonists
    Pinzani, D
    Papini, AM
    Vallecchi, ME
    Chelli, M
    Ginanneschi, M
    Rapi, G
    Quartara, L
    Patacchini, R
    Maggi, CA
    Arcamone, FM
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1996, 6 (04) : 367 - 372
  • [5] DUAL ANTAGONISTS FOR NK1 AND NK2 RECEPTORS SHOWING INVITRO AND INVIVO SPECIES SELECTIVITY FOR TACHYKININ RECEPTORS
    ROBINEAU, P
    LONCHAMPT, M
    KUCHARCZYK, N
    KRAUSE, JE
    BATAILLE, I
    GAUDIN, M
    SICOT, N
    TISSERAND, F
    FAUCHERE, JL
    CANET, E
    AMERICAN REVIEW OF RESPIRATORY DISEASE, 1993, 147 (04): : A709 - A709
  • [6] NEW SPIROPIPERIDINES AS POTENT AND SELECTIVE NONPEPTIDE TACHYKININ NK2 RECEPTOR ANTAGONISTS
    SMITH, PW
    COOPER, AWJ
    BELL, R
    BERESFORD, IJM
    GORE, PM
    MCELROY, AB
    PRITCHARD, JM
    SAEZ, V
    TAYLOR, NR
    SHELDRICK, RLG
    WARD, P
    JOURNAL OF MEDICINAL CHEMISTRY, 1995, 38 (19) : 3772 - 3779
  • [7] PEPTIDE-BASED TACHYKININ NK2 RECEPTOR ANTAGONISTS
    QUARTARA, L
    ROVERO, P
    MAGGI, CA
    MEDICINAL RESEARCH REVIEWS, 1995, 15 (02) : 139 - 155
  • [8] 2 NONPEPTIDE TACHYKININ ANTAGONISTS ACT THROUGH EPITOPES ON CORRESPONDING SEGMENTS OF THE NK1 AND NK2 RECEPTORS
    GETHER, U
    YOKOTA, Y
    EMONDSALT, X
    BRELIERE, JC
    LOWE, JA
    SNIDER, RM
    NAKANISHI, S
    SCHWARTZ, TW
    PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1993, 90 (13) : 6194 - 6198
  • [9] Mutagenesis at the human tachykinin NK2 receptor to define the binding site of a novel class of antagonists
    Meini, S
    Bellucci, F
    Catalani, C
    Cucchi, P
    Patacchini, R
    Rotondaro, L
    Altamura, M
    Giuliani, S
    Giolitti, A
    Maggi, CA
    EUROPEAN JOURNAL OF PHARMACOLOGY, 2004, 488 (1-3) : 61 - 69
  • [10] Discovery of a new series of potent and selective linear tachykinin NK2 receptor antagonists
    Fedi, Valentina
    Altamura, Maria
    Catalioto, Rose-Marie
    Giannotti, Danilo
    Giolitti, Alessandro
    Giuliani, Sandro
    Guidi, Antonio
    Harmat, Nicholas J. S.
    Lecci, Alessandro
    Meini, Stefania
    Nannicini, Rossano
    Pasqui, Franco
    Tramontana, Manuela
    Triolo, Antonio
    Maggi, Carlo Alberto
    JOURNAL OF MEDICINAL CHEMISTRY, 2007, 50 (20) : 4793 - 4807