STRUCTURE-ACTIVITY RELATIONS IN AUREOLIC ACID GROUP OF ANTIBIOTICS - COMPLEX-FORMATION WITH DNA AND INHIBITION OF RNA-SYNTHESIS

被引：0
|
作者：
KISELEVA, OA [1 ]
VOLKOVA, NG [1 ]
STUKACHEVA, EA [1 ]
SHEMYAKIN, MF [1 ]
BERLIN, YA [1 ]
KOLOSOV, MN [1 ]
机构：
[1] MM SHEMYAKINA NAT PROD CHEM INST, MOSCOW, USSR
来源：
MOLEKULYARNAYA BIOLOGIYA | 1973年 / 7卷 / 06期
关键词：
D O I：
暂无
中图分类号：
Q5 [生物化学]; Q7 [分子生物学];
学科分类号：
071010 ; 081704 ;
摘要：
引用
收藏
页码：900 / 907
页数：8
相关论文
共 43 条
  • [31] 2-methoxyestradiol and analogs as novel antiproliferative agents: Analysis of three-dimensional quantitative structure-activity relationships for DNA synthesis inhibition and estrogen receptor binding
    Hughes, RA
    Harris, T
    Altmann, E
    McAllister, D
    Vlahos, R
    Robertson, A
    Cushman, M
    Wang, ZQ
    Stewart, AG
    MOLECULAR PHARMACOLOGY, 2002, 61 (05) : 1053 - 1069
  • [32] Dimeric 1,3-Phenylene-bis(piperazinyl benzimidazole)s: Synthesis and Structure-Activity Investigations on their Binding with Human Telomeric G-Quadruplex DNA and Telomerase Inhibition Properties
    Jain, Akash K.
    Paul, Ananya
    Maji, Basudeb
    Muniyappa, K.
    Bhattacharya, Santanu
    JOURNAL OF MEDICINAL CHEMISTRY, 2012, 55 (07) : 2981 - 2993
  • [33] Synthesis, crystal structure and antiproliferative activity of Cu(II) nalidixic acid-DACH conjugate: Comparative in vitro DNA/RNA binding profile, cleavage activity and molecular docking studies
    Arjmand, Farukh
    Yousuf, Imtiyaz
    ben Hadda, Taibi
    Toupet, Loic
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2014, 81 : 76 - 88
  • [34] Facile one-pot synthesis, butyrylcholinesterase and α-glucosidase inhibitory activities, structure-activity relationship, molecular docking and DNA-drug binding analysis of Meldrum's acid derivatives
    Mehfooz, Haroon
    Saeed, Aamer
    Faisal, Muhammad
    Larik, Fayaz Ali
    Muqadar, Urooj
    Khatoon, Saira
    Channar, Pervaiz Ali
    Ismail, Hammad
    Bilquees, Salma
    Bashid, Sajid
    Shafique, Shagufta
    Mirza, Bushra
    Dilshad, Erum
    Ahmad, Fawad
    RESEARCH ON CHEMICAL INTERMEDIATES, 2020, 46 (05) : 2437 - 2456
  • [35] Discovery, synthesis, and structure-activity relations of 3,4-dihydro-1H-spiro(naphthalene-2,2′-piperidin)-1-ones as potassium-competitive acid blockers
    Imaeda, Toshihiro
    Ono, Koji
    Nakai, Kazuo
    Hori, Yasunobu
    Matsukawa, Jun
    Takagi, Terufumi
    Fujioka, Yasushi
    Tarui, Naoki
    Kondo, Mitsuyo
    Imanishi, Akio
    Inatomi, Nobuhiro
    Kajino, Masahiro
    Itoh, Fumio
    Nishida, Haruyuki
    BIOORGANIC & MEDICINAL CHEMISTRY, 2017, 25 (14) : 3719 - 3735
  • [36] Synthesis, crystal structure, antimicrobial activity and DNA-binding of hydrogen-bonded proton-transfer complex of 2,6-diaminopyridine with picric acid
    Khan, Ishaat M.
    Ahmad, Afaq
    Ullah, M. F.
    JOURNAL OF PHOTOCHEMISTRY AND PHOTOBIOLOGY B-BIOLOGY, 2011, 103 (01) : 42 - 49
  • [37] Inhibition of secretory phospholipase A2.: 1-Design, synthesis and structure-activity relationship studies starting from 4-tetradecyloxybenzamidine to obtain specific inhibitors of group II sPLA2s
    Assogba, L
    Ahamada-Himidi, A
    Habich, NMB
    Aoun, D
    Boukli, L
    Massicot, F
    Mounier, CM
    Huet, J
    Lamouri, A
    Ombetta, JE
    Godfroid, JJ
    Dong, CZ
    Heymans, F
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2005, 40 (09) : 850 - 861
  • [38] Resistance-modifying agents.: 11.: Pyrimido[5,4-d]pyrimidine modulators of antitumor drug activity.: Synthesis and structure-activity relationships for nucleoside transport inhibition and binding to α1-acid glycoprotein
    Curtin, NJ
    Barlow, HC
    Bowman, KJ
    Calvert, AH
    Davison, R
    Golding, BT
    Huang, B
    Loughlin, PJ
    Newell, DR
    Smith, PG
    Griffin, RJ
    JOURNAL OF MEDICINAL CHEMISTRY, 2004, 47 (20) : 4905 - 4922
  • [39] Structure-activity relationship of a series of C-terminus modified aminoalkyl, diaminoalkyl- and anilino-containing analogues of the benzoic acid mustard distamycin derivative tallimustine: Synthesis, DNA binding and cytotoxicity studies
    Brooks, N
    Hartley, JA
    Simpson, JE
    Wright, SR
    Woo, S
    Centioni, S
    Fontaine, MD
    McIntyre, TE
    Lee, M
    BIOORGANIC & MEDICINAL CHEMISTRY, 1997, 5 (08) : 1497 - 1507
  • [40] Synthesis, in vitro pharmacology, structure-activity relationships, and pharmacokinetics of 3-alkoxy-2-amino-6-fluorobicyclo[3.1.0]hexane-2,6-dicarboxylic acid derivatives as potent and selective group II metabotropic glutamate receptor antagonists
    Nakazato, A
    Sakagami, K
    Yasuhara, A
    Ohta, H
    Yoshikawa, R
    Itoh, M
    Nakamura, M
    Chaki, S
    JOURNAL OF MEDICINAL CHEMISTRY, 2004, 47 (18) : 4570 - 4587
12345