BINDING OF THE BOVINE BASIC PANCREATIC TRYPSIN-INHIBITOR (KUNITZ) TO HUMAN ALPHA-THROMBIN, BETA-THROMBIN AND GAMMA-THROMBIN - A KINETIC AND THERMODYNAMIC STUDY

被引:27
|
作者
ASCENZI, P
COLETTA, M
AMICONI, G
DECRISTOFARO, R
BOLOGNESI, M
GUARNERI, M
MENEGATTI, E
机构
[1] CATHOLIC UNIV ROME, INST CHEM, ROME, ITALY
[2] UNIV PAVIA, DEPT GENET & MICROBIOL, CRYSTALLOG SECT, I-27100 PAVIA, ITALY
[3] UNIV FERRARA, DEPT PHARMACEUT SCI, I-44100 FERRARA, ITALY
关键词
D O I
10.1016/0167-4838(88)90262-2
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:156 / 161
页数:6
相关论文
共 47 条
  • [31] BINDING OF PORCINE PANCREATIC SECRETORY TRYPSIN-INHIBITOR TO BOVINE BETA-TRYPSIN - A KINETIC-STUDY
    ASCENZI, P
    AMICONI, G
    BOLOGNESI, M
    MENEGATTI, E
    GUARNERI, M
    BIOPOLYMERS, 1986, 25 (12) : 2325 - 2333
  • [32] First complex of human alpha-thrombin to crystallographic and kinetic analysis and evidence of binding mechanism
    Shordalakes, E
    Green, D
    Merette, S
    Goodwin, CA
    Scully, MF
    Dodson, G
    Kakkar, VV
    Deadman, JJ
    THROMBOSIS AND HAEMOSTASIS, 1999, : 703 - 703
  • [33] COVALENT STRUCTURES OF THE AUTOLYTIC BETA-DERIVATIVES AND GAMMA-DERIVATIVES OF HUMAN ALPHA-THROMBIN
    BOISSEL, JP
    RABIET, MJ
    LABIE, D
    ELION, J
    THROMBOSIS AND HAEMOSTASIS, 1983, 50 (01) : 265 - 265
  • [34] TRANSIENT REMOVAL OF PROFLAVINE INHIBITION OF BOVINE BETA-TRYPSIN BY THE BOVINE BASIC PANCREATIC TRYPSIN-INHIBITOR (KUNITZ) - A CASE FOR CHRONOSTERIC EFFECTS
    ANTONINI, E
    ASCENZI, P
    BOLOGNESI, M
    MENEGATTI, E
    GUARNERI, M
    JOURNAL OF BIOLOGICAL CHEMISTRY, 1983, 258 (08) : 4676 - 4678
  • [35] Mutations within the reactive-site region of human pancreatic secretory trypsin inhibitor confer alpha-thrombin and factor Xa inhibitory activities
    Katoh, T
    Tamaki, M
    Kikuchi, N
    Teraoka, H
    Nagata, K
    Yoshida, N
    BIOSCIENCE BIOTECHNOLOGY AND BIOCHEMISTRY, 1997, 61 (02) : 389 - 391
  • [36] GLU(192)-]GLN SUBSTITUTION IN THROMBIN YIELDS AN ENZYME THAT IS EFFECTIVELY INHIBITED BY BOVINE PANCREATIC TRYPSIN-INHIBITOR AND TISSUE FACTOR PATHWAY INHIBITOR
    GUINTO, ER
    YE, J
    LEBONNIEC, BF
    ESMON, CT
    JOURNAL OF BIOLOGICAL CHEMISTRY, 1994, 269 (28) : 18395 - 18400
  • [37] INHIBITION OF BOVINE BETA-TRYPSIN, HUMAN ALPHA-THROMBIN AND PORCINE PANCREATIC BETA-KALLIKREIN-B BY BENZAMIDINE AND ITS BIS-DERIVATIVES, TRIS-DERIVATIVES AND TETRA-DERIVATIVES - THERMODYNAMIC AND MOLECULAR MODELING STUDY
    MENEGATTI, E
    FERRONI, R
    NASTRUZZI, C
    BORTOLOTTI, F
    SCALIA, S
    AMICONI, G
    BOLOGNESI, M
    COLETTA, M
    ONESTI, S
    FRUTTERO, R
    ASCENZI, P
    FARMACO, 1991, 46 (11): : 1297 - 1310
  • [38] EFFECT OF HUMAN ALPHA-THROMBIN ON THE TRANSFORMING GROWTH FACTOR-BETA-1-BINDING ACTIVITY OF HUMAN ALPHA-2-MACROGLOBULIN
    WEBB, DJ
    LAMARRE, J
    GONIAS, SL
    SEMINARS IN THROMBOSIS AND HEMOSTASIS, 1992, 18 (03): : 305 - 310
  • [39] INHIBITION OF BOVINE BETA-TRYPSIN, HUMAN ALPHA-THROMBIN AND PORCINE PANCREATIC BETA-KALLIKREIN-B BY 4',6-DIAMIDINO-2-PHENYLINDOLE, 6-AMIDINOINDOLE AND BENZAMIDINE - A COMPARATIVE THERMODYNAMIC AND X-RAY STRUCTURAL STUDY
    CASALE, E
    COLLYER, C
    ASCENZI, P
    BALLIANO, G
    MILLA, P
    VIOLA, F
    FASANO, M
    MENEGATTI, E
    BOLOGNESI, M
    BIOPHYSICAL CHEMISTRY, 1995, 54 (01) : 75 - 81
  • [40] CATALYTIC PROPERTIES OF SERINE PROTEASES .2. COMPARISON BETWEEN HUMAN URINARY KALLIKREIN AND HUMAN UROKINASE, BOVINE BETA-TRYPSIN, BOVINE THROMBIN, AND BOVINE ALPHA-CHYMOTRYPSIN
    ASCENZI, P
    MENEGATTI, E
    GUARNERI, M
    BORTOLOTTI, F
    ANTONINI, E
    BIOCHEMISTRY, 1982, 21 (10) : 2483 - 2490