ASYMMETRIC-SYNTHESIS OF (3S)-2,3,4,5-TETRAHYDROPYRIDAZINE-3-CARBOXYLIC ACID

被引：43
|
作者：
ASPINALL, IH
COWLEY, PM
MITCHELL, G
STOODLEY, RJ
机构：
[1] UMIST,DEPT CHEM,POB 88,MANCHESTER M60 1QD,ENGLAND
[2] ZENECA AGROCHEM,JEALOTTS HILL RES STN,BRACKNELL RG12 6EY,BERKS,ENGLAND
来源：
JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS | 1993年 / 15期
关键词：
D O I：
10.1039/c39930001179
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
The title compound 1a is prepared by a two-step sequence from the cycloadduct 5d, derived from di(tert-butyl) azodicarboxylate and the diene 4b by a hetero Diels-Alder reaction.
引用
收藏
页码：1179 / 1180
页数：2
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