N-(INDOL-3-YLGLYOXYLYL)AMINO ACID ESTER DERIVATIVES - SYNTHESIS AND INTERACTION PROPERTIES AT THE BENZODIAZEPINE RECEPTOR

被引：0

作者：

PRIMOFIORE, G ^{[1
]}

DASETTIMO, F ^{[1
]}

MARINI, AM ^{[1
]}

LAMOTTA, C ^{[1
]}

MARTINI, C ^{[1
]}

SENATORE, G ^{[1
]}

LUCACCHINI, A ^{[1
]}

机构：

[1] UNIV PISA, IST POLICATTEDRA DISCIPLINE BIOL, I-56126 PISA, ITALY

来源：

FARMACO | 1995年 / 50卷 / 01期

关键词：

D O I：

暂无

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

Several N-(indol-3-ylglyoxylyl)alanine and glycine ester derivatives were prepared to evaluate the influence of the ester group size both on affinity and on activity at the benzodiazepine receptor. Moreover, indol-3-ylglyoxylic acid esters, closely related to 3-alkoxy-beta-carbolines, were synthesized and tested in vitro on the benzodiazepine receptor.

引用

页码：5 / 12

页数：8

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