PREPARATION OF 3,6-DIHYDRO-2H-1,3-OXAZINES AND THEIR USE AS POTENTIAL 1,3-AMINO ALCOHOL SYNTHONS

被引：0

作者：

CHERKAUSKAS, JP ^{[1
]}

BORZILLERI, RM ^{[1
]}

SISKO, J ^{[1
]}

WEINREB, SM ^{[1
]}

机构：

[1] PENN STATE UNIV,DEPT CHEM,UNIVERSITY PK,PA 16802

来源：

SYNLETT | 1995年 / 05期

关键词：

N-SULFINYL-P-TOLUENESULFONAMIDE; BETA-HYDROXYALDEHYDES TETRAHYDRO-1,3-OXAZINES;

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

3,6-Dihydro-2H-1,3-oxazines, which can be readily prepared by reaction of beta-hydroxyaldehydes with N-sulfinyl-p-toluenesulfonamide, are useful intermediates for stereoselective synthesis of 1,3-amino alcohol derivatives.

引用

页码：527 / 528

页数：2

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