SYNTHESIS OF 3-(1,2,3,6-TETRAHYDRO PYRIDIN-4-YL) 1H-INDOLES AND STUDY OF THEIR SEROTONINERGIC AND ANTIDOPAMINERGIC PROPERTIES

被引：45
|
作者：
GUILLAUME, J [1 ]
DUMONT, C [1 ]
LAURENT, J [1 ]
NEDELEC, L [1 ]
机构：
[1] ROUSSEL UCLAF,CTR RECH,102 ROUTE NOISY,F-93230 ROMAINVILLE,FRANCE
来源：
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | 1987年 / 22卷 / 01期
关键词：
D O I：
10.1016/0223-5234(87)90172-3
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
引用
收藏
页码：33 / 43
页数：11
相关论文
共 50 条
  • [21] Facile and Efficient Synthesis of Ethyl 3-oxo-3-(pyridin-4-yl)-2-((pyridin-4-yl)methylene)propanoate
    Erenler, Ramazan
    ASIAN JOURNAL OF CHEMISTRY, 2011, 23 (08) : 3763 - 3764
  • [22] The crystal structure of hexaqua(μ2-3-(3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl)propanoato-1κ2O,O′; 2κO′)(3-(3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl)propanoato-κO)(3-(3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl)propanoato-κ2O,O′) digadolinium(III)octahydrate, C60H76Gd2N18O32
    Chen, Qifan
    Huang, Fang
    Quan, Wenjing
    Lu, Yanhua
    Zhang, Fang
    Liu, Fei
    ZEITSCHRIFT FUR KRISTALLOGRAPHIE-NEW CRYSTAL STRUCTURES, 2016, 231 (02): : 457 - 460
  • [23] Synthesis and characterization of a pegylated derivative of 3-(1,2,3,6-tetrahydro-pyridin-4yl)-1H-indole (IDT199): A high affinity SERT ligand for conjugation to quantum dots
    Tomlinson, Ian D.
    Warnerment, Michael R.
    Mason, John N.
    Vergne, Matthew J.
    Hercules, David M.
    Blakely, Randy D.
    Rosenthal, Sandra J.
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2007, 17 (20) : 5656 - 5660
  • [24] 2-(Pyridin-4-yl)-1H-benzimidazole
    Geiger, David K.
    Bond, Christopher J.
    ACTA CRYSTALLOGRAPHICA SECTION E-CRYSTALLOGRAPHIC COMMUNICATIONS, 2013, 69 : O869 - +
  • [25] Synthesis,Crystal Structure and Fluorescent Properties of a Cadmium(Ⅱ) Complex with 3-(Pyridin-4-yl)-5-(pyrazin-2-yl)-1H-1,2,4-triazole
    王玉芳
    孙小媛
    耿俊磊
    结构化学, 2016, 35 (03) : 397 - 403
  • [26] A convenient synthesis of 3-substituted 1H-indoles
    Technical R and D, Sandoz Research Institute, Sandoz Pharmaceutical Corporation, East Hanover, NJ 07936, United States
    SYNTH. COMMUN., 1 (95-100):
  • [27] 4-[3-(Pyridin-4-yl)propyl]pyridinium 2-carboxybenzoate
    Xu, Wei
    Qi, Jin-Li
    ACTA CRYSTALLOGRAPHICA SECTION E-CRYSTALLOGRAPHIC COMMUNICATIONS, 2012, 68 : 02319 - +
  • [28] 4-[(3-Nitrobenzylidene)amino]-3-(pyridin-4-yl)-1H-1,2,4-triazole-5(4H)-thione
    Li, Tian-Bao
    Yang, Ming-Sheng
    Yin, Bang-Shao
    ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE, 2012, 68 : O279 - U1635
  • [29] A CONVENIENT SYNTHESIS OF 3-SUBSTITUTED 1H-INDOLES
    PRASHAD, M
    LAVECCHIA, L
    PRASAD, K
    REPIC, O
    SYNTHETIC COMMUNICATIONS, 1995, 25 (01) : 95 - 100
  • [30] Synthesis of E/Z 3-(1H-benzotriazol-1-yl)-3-(pyridin-4-yl)acrylonitriles and E/Z 2-(3-imino-2-benzofuran-1(3H)ylidene)acetonitriles.: An unusual case of displacement of the benzotriazole ring
    Carta, A
    Sanna, P
    Bacchi, A
    HETEROCYCLES, 2002, 57 (06) : 1079 - 1090
12345