EVALUATION OF A NOVEL ORALLY-ACTIVE DIRECT INHIBITOR OF THROMBIN IN ANIMAL-MODELS OF THROMBOSIS

被引:0
|
作者
ROTE, WE [1 ]
DEMPSEY, EM [1 ]
OLDESCHULTE, GL [1 ]
ARDECKY, RJ [1 ]
TAMURA, SY [1 ]
NUTT, RF [1 ]
BERGUM, PW [1 ]
TRAN, HS [1 ]
ANDERSON, SM [1 ]
VLASUK, GP [1 ]
机构
[1] CORVAS INT INC,SAN DIEGO,CA
关键词
D O I
暂无
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
引用
收藏
页码:344 / 344
页数:1
相关论文
共 50 条
  • [31] ANIMAL-MODELS IN THE EVALUATION OF ANTIMICROBIAL AGENTS
    ZAK, O
    OREILLY, T
    ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 1991, 35 (08) : 1527 - 1531
  • [32] FK-906, A HIGHLY POTENT, ORALLY-ACTIVE HUMAN RENIN INHIBITOR
    NEYA, M
    MARUSAWA, H
    IMAL, K
    KAYAKIRI, N
    WATANABE, S
    HEMML, K
    HASHIMOTO, M
    TANAKA, H
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1993, 206 : 56 - MEDI
  • [33] ANIMAL-MODELS - THE INVIVO EVALUATION OF CIPROFLOXACIN
    PETERSON, LR
    JOURNAL OF ANTIMICROBIAL CHEMOTHERAPY, 1986, 18 : 55 - 64
  • [34] ANTITHROMBOTIC ACTIVITY OF RPR110173, AN ORALLY-ACTIVE PLATELET FIBRINOGEN RECEPTOR ANTAGONIST, IN CANINE MODELS OF ARTERIAL THROMBOSIS
    LEADLEY, RJ
    BOSTWICK, JS
    KASIEWSKI, CJ
    CHU, V
    KLEIN, SI
    CZEKAJ, M
    GARDNER, CJ
    PERRONE, MH
    DUNWIDDIE, CT
    CIRCULATION, 1995, 92 (08) : 2329 - 2329
  • [35] MACROCYCLIC RENIN INHIBITORS - SYNTHESIS OF A SUBNANOMOLAR, ORALLY-ACTIVE CYSTEINE DERIVED INHIBITOR
    YANG, LH
    WEBER, AE
    GREENLEE, WJ
    PATCHETT, AA
    TETRAHEDRON LETTERS, 1993, 34 (44) : 7035 - 7038
  • [36] DESIGN AND SYNTHESIS OF AN ORALLY-ACTIVE MACROCYCLIC NEUTRAL ENDOPEPTIDASE-24.11 INHIBITOR
    MACPHERSON, LJ
    BAYBURT, EK
    CAPPARELLI, MP
    BOHACEK, RS
    CLARKE, FH
    GHAI, RD
    SAKANE, Y
    BERRY, CJ
    PEPPARD, JV
    TRAPANI, AJ
    JOURNAL OF MEDICINAL CHEMISTRY, 1993, 36 (24) : 3821 - 3828
  • [37] LB30057, an orally effective direct thrombin inhibitor, prevents arterial and venous thrombosis in Rats and Dogs
    Hee Dong Park
    Hee Jin Kim
    Yeong Soo Oh
    In Chull Kim
    Yong Zu Kim
    Hyun Chul Koh
    In Chul Shin
    Yong Hee Lee
    Chang Ho Lee
    Archives of Pharmacal Research, 2003, 26 : 224 - 231
  • [38] LB30057, an orally effective direct thrombin inhibitor, prevents arterial and venous thrombosis in rats and dogs
    Park, HD
    Kim, HJ
    Oh, YS
    Kim, IC
    Kim, YZ
    Koh, HC
    Shin, IC
    Lee, YH
    Lee, CH
    ARCHIVES OF PHARMACAL RESEARCH, 2003, 26 (03) : 224 - 231
  • [39] A novel inhibitor of activated thrombin activatable fibrinolysis inhibitor (TAFIa) - Part II: Enhancement of both exogenous and endogenous fibrinolysis in animal models of thrombosis
    Wang, Yi-Xin
    da Cunha, Valcleci
    Vincelette, Jon
    Zhao, Lei
    Nagashima, Mariko
    Kawai, Kohichi
    Yuan, Shendong
    Emayan, Kumar
    Islam, Imadul
    Hosoya, Junko
    Sullivan, Mark E.
    Dole, William P.
    Morser, John
    Buckman, Brad O.
    Vergona, Ronald
    THROMBOSIS AND HAEMOSTASIS, 2007, 97 (01) : 54 - 61
  • [40] UK-14,275, A NOVEL ORALLY-ACTIVE CARDIAC STIMULANT
    ALABASTER, CT
    BLACKBURN, KJ
    JOICE, JR
    MASSINGHAM, R
    SCHOLFIELD, PC
    BRITISH JOURNAL OF PHARMACOLOGY, 1977, 60 (02) : 284 - 285