DIURETICS .4. 6-CHLORO-3-SUBSTITUTED 7-SULFAMOYL-1,2,4-BENZOTHIADIAZINE 1,1-DIOXIDES

被引:13
|
作者
WHITEHEAD, C
TRAVERSO, JJ
MORRISON, DE
MARSHALL, FJ
机构
来源
JOURNAL OF ORGANIC CHEMISTRY | 1961年 / 26卷 / 08期
关键词
D O I
10.1021/jo01066a045
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
引用
收藏
页码:2809 / &
相关论文
共 50 条
  • [41] New substituted aryl esters and aryl amides of 3,4-dihydro-2H-1,2,4-benzothiadiazine 1,1-dioxides as positive allosteric modulators of AMPA receptors
    Dintilhac, Gaeelle
    Arslan, Deniz
    Dilly, Sebastien
    Danober, Laurence
    Botez, Iuliana
    Lestage, Pierre
    Pirotte, Bernard
    de Tullio, Pascal
    MEDCHEMCOMM, 2011, 2 (06) : 509 - 523
  • [42] CORRELATION OF ANTIHYPERTENSIVE ACTIVITY WITH STRUCTURE IN A SERIES OF 2H-1,2,4-BENZOTHIADIAZINE 1,1-DIOXIDES USING SUBSTITUENT CONSTANT APPROACH
    TOPLISS, JG
    YUDIS, MD
    JOURNAL OF MEDICINAL CHEMISTRY, 1972, 15 (04) : 394 - &
  • [43] 7-Iodo-3-isopropylamino-4H-1,2,4-benzothiadiazine 1,1-dioxide
    Unité de Cristallographie, Institut de Physique B5, Univ. de Liege au Sart Tilman, B-4000 Liège, Belgium
    不详
    Acta Crystallogr Sect C Cryst Struct Commun, 7 (1152-1154):
  • [44] Triphenylphosphonium salts of 1,2,4-benzothiadiazine 1,1-dioxides related to diazoxide targeting mitochondrial ATP-sensitive potassium channels
    Constant-Urban, Celine
    Charif, Mounia
    Goffin, Eric
    Van Heugen, Jean-Claude
    Elmoualij, Benaissa
    Chiap, Patrice
    Mouithys-Mickalad, Ange
    Serteyn, Didier
    Lebrun, Philippe
    Pirotte, Bernard
    De Tullio, Pascal
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2013, 23 (21) : 5878 - 5881
  • [45] Chloro-Substituted 3-Alkylamino-4H-1,2,4-benzothiadiazine 1,1-Dioxides as ATP-Sensitive Potassium Channel Activators: Impact of the Position of the Chlorine Atom on the Aromatic Ring on Activity and Tissue Selectivity
    Pirotte, Bernard
    de Tullio, Pascal
    Nguyen, Quynh-Anh
    Somers, Fabian
    Fraikin, Pierre
    Florence, Xavier
    Wahl, Philip
    Hansen, John Bondo
    Lebrun, Philippe
    JOURNAL OF MEDICINAL CHEMISTRY, 2010, 53 (01) : 147 - 154
  • [46] MASS-SPECTROMETRIC FRAGMENTATION PATTERNS OF SOME BIOLOGICALLY-ACTIVE DERIVATIVES OF 2H-1,2,4-BENZOTHIADIAZINE 1,1-DIOXIDES
    KIRKIENRZESZOTA.AM
    PLIMMER, JR
    KREES, SV
    RZESZOTARSKI, WJ
    JOURNAL OF HETEROCYCLIC CHEMISTRY, 1975, 12 (01) : 155 - 159
  • [47] Synthesis of 3-substituted 4,1,2-benzothiadiazine 4,4-dioxides and 2 or 3-substituted 1,4-benzothiazine 1,1-dioxides
    Balbi, A
    Sottofattori, E
    Mazzei, M
    JOURNAL OF HETEROCYCLIC CHEMISTRY, 1996, 33 (02) : 347 - 350
  • [48] Toward tissue-selective pancreatic B-cells KATP channel openers belonging to 3-alkylamino-7-halo-4H-1,2,4-benzothiadiazine 1,1-dioxides
    de Tullio, P
    Becker, B
    Boverie, S
    Dabrowski, M
    Wahl, P
    Antoine, MH
    Somers, F
    Sebille, S
    Ouedraogo, R
    Hansen, JB
    Lebrun, P
    Pirotte, B
    JOURNAL OF MEDICINAL CHEMISTRY, 2003, 46 (15) : 3342 - 3353
  • [49] ANTIBACTERIAL ACTIVITY AND SYNTHESES OF 4-(SUBSTITUTED BENZYLAMINO)-1,2,3-BENZOTHIADIAZINE-1,1-DIOXIDES
    SADANA, GS
    PRADHAN, NS
    DEODHAR, KD
    INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY, 1990, 29 (06): : 598 - 599
  • [50] 3-Alkylamino-4H-1,2,4-benzothiadiazine 1,1-dioxides as ATP-sensitive potassium channel openers:: Effect of 6,7-disubstitution on potency and tissue selectivity
    de Tullio, P
    Boverie, S
    Becker, B
    Antoine, MH
    Nguyen, QA
    Francotte, P
    Counerotte, S
    Sebille, S
    Pirotte, B
    Lebrun, P
    JOURNAL OF MEDICINAL CHEMISTRY, 2005, 48 (15) : 4990 - 5000