A STEREOCONTROLLED SYNTHESIS OF HYDROXYETHYLENE DIPEPTIDE ISOSTERES USING NOVEL, CHIRAL AMINOALKYL EPOXIDES AND GAMMA-(AMINOALKYL) GAMMA-LACTONES

被引：153

作者：

EVANS, BE ^{[1
]}

RITTLE, KE ^{[1
]}

HOMNICK, CF ^{[1
]}

SPRINGER, JP ^{[1
]}

HIRSHFIELD, J ^{[1
]}

VEBER, DF ^{[1
]}

机构：

[1] MERCK INST THERAPEUT RES,RAHWAY,NJ 07065

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1985年 / 50卷 / 23期

关键词：

D O I：

10.1021/jo00223a037

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

页码：4615 / 4625

页数：11

共 42 条

[1] AN EFFICIENT SYNTHESIS OF GAMMA-LACTONES AS PRECURSORS OF HYDROXYETHYLENE DIPEPTIDE ISOSTERE
SAKURAI, M
SAITO, F
OHATA, Y
YABE, Y
NISHI, T
JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS, 1992, (21) : 1562 - 1563
[2] NEW DIASTEREOSELECTIVE SYNTHESIS OF NOVEL CHIRAL GAMMA-(AMINOALKYL)-ALPHA-HYDROXY-GAMMA-LACTONES AND THEIR APPLICATION FOR THE SYNTHESIS OF RENIN INHIBITORS
METTERNICH, R
LUDI, W
TETRAHEDRON LETTERS, 1988, 29 (32) : 3923 - 3926
[3] AN APPROACH TO THE STEREOCONTROLLED SYNTHESIS OF POLYSUBSTITUTED CHIRAL BUTENOLIDES AND GAMMA-LACTONES
RODRIGUEZ, CM
MARTIN, VS
TETRAHEDRON LETTERS, 1991, 32 (19) : 2165 - 2168
[4] LACTONES .3. SYNTHESIS OF ALPHA-AMINOALKYL-GAMMA-LACTONES
LEHMANN, J
REUSCH, T
ARCHIV DER PHARMAZIE, 1983, 316 (11) : 955 - 960
[5] LACTONES .4. SYNTHESIS OF DIHYDROXYLATED DIPHENYLALKANAMINES VIA AMINOALKYL-GAMMA-LACTONES
LEHMANN, J
ARCHIV DER PHARMAZIE, 1984, 317 (02) : 126 - 133
[6] SYNTHESIS AND STEREOCHEMISTRY OF NOVEL TRICYCLIC GAMMA-LACTONES
VASSILEV, V
BLAGOEV, B
BULLETIN DE LA SOCIETE CHIMIQUE DE FRANCE, 1991, (04): : 525 - 529
[7] A CONVENIENT SYNTHESIS OF SUBSTITUTED CHIRAL TETRAHYDROFURANS FROM SUGAR GAMMA-LACTONES
CHAPLEUR, Y
JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS, 1984, (07) : 449 - 450
[8] A NOVEL SYNTHESIS OF ERITADENINE - REACTIONS OF SOME PURINES WITH GAMMA-LACTONES
OKUMURA, K
OINE, T
YAMADA, Y
TOMIE, M
NAGURA, T
KAWAZU, M
MIZOGUCH.T
INOUE, I
JOURNAL OF THE CHEMICAL SOCIETY D-CHEMICAL COMMUNICATIONS, 1970, (17): : 1045 - &
[9] AN EFFICIENT SYNTHESIS OF THE GAMMA-LACTONE CORRESPONDING TO A HYDROXYETHYLENE DIPEPTIDE ISOSTERE USING STEREOSELECTIVE BROMOLACTONIZATION OF A CHIRAL ACYLOXAZOLIDINONE
BRADBURY, RH
REVILL, JM
RIVETT, JE
WATERSON, D
TETRAHEDRON LETTERS, 1989, 30 (29) : 3845 - 3848
[10] Synthesis of functionalized gamma- and delta-lactones via polymer-bound epoxides
LeHetet, C
David, M
Carreaux, F
Carboni, B
Sauleau, A
TETRAHEDRON LETTERS, 1997, 38 (29) : 5153 - 5156

← 1 2 3 4 5 →