SPECIFIC HIV-1 REVERSE-TRANSCRIPTASE INHIBITORS

被引:16
|
作者
DEBYSER, Z
PAUWELS, R
ANDRIES, K
DE CLERCQ, E
机构
[1] CATHOLIC UNIV LEUVEN, REGA INST MED RES, B-3000 LOUVAIN, BELGIUM
[2] JANSSEN RES FDN, B-2340 BEERSE, BELGIUM
来源
JOURNAL OF ENZYME INHIBITION | 1992年 / 6卷 / 01期
关键词
HIV-1; REVERSE TRANSCRIPTASE; INHIBITORS; AZT; HEPT; TIBO;
D O I
10.3109/14756369209041355
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
[No abstract available]
引用
下载
收藏
页码:47 / 53
页数:7
相关论文
共 50 条
  • [31] DISCOVERY AND DESIGN OF POTENT BISHETEROARYLPIPERAZINE (BHAP) HIV-1 REVERSE-TRANSCRIPTASE INHIBITORS
    ROMERO, DL
    THOMAS, RC
    MORGE, RA
    POEL, TJ
    HOSLEY, MJ
    PALMER, JR
    ARISTOFF, PA
    JOHNSON, PD
    REUSSER, F
    ALTHAUS, IW
    TARPLEY, WG
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1992, 204 : 134 - MEDI
  • [32] INHIBITORS OF HIV-1 REVERSE-TRANSCRIPTASE AND FIDELITY OF INVITRO DNA-REPLICATION
    ABBOTTS, J
    WILSON, SH
    JOURNAL OF ENZYME INHIBITION, 1992, 6 (01): : 35 - 46
  • [33] STRUCTURE-ACTIVITY STUDIES OF NOVEL INHIBITORS OF HIV-1 REVERSE-TRANSCRIPTASE
    LYLE, TA
    YOUNG, SD
    ANDERSON, PS
    BALANI, SK
    BRITCHER, SF
    CARROLL, SS
    CULBERSON, C
    EMINI, EA
    GOLDMAN, ME
    HOMNICK, CF
    HUFF, JR
    LUMMA, WC
    OBRIEN, JA
    OLSEN, DB
    PAYNE, LS
    PETTIBONE, DJ
    QUINTERO, JC
    SANDERS, WM
    SANDERSON, PEJ
    SCHLEIF, WA
    SMITH, SJ
    STAHLHUT, M
    THEOHARIDES, AM
    THOMAS, CM
    TRAN, LO
    TUCKER, TJ
    WISCOUNT, CM
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1993, 206 : 135 - MEDI
  • [34] HIV RESISTANCE TO REVERSE-TRANSCRIPTASE INHIBITORS
    DECLERCQ, E
    BIOCHEMICAL PHARMACOLOGY, 1994, 47 (02) : 155 - 169
  • [35] HIV INHIBITORS TARGETED AT THE REVERSE-TRANSCRIPTASE
    DECLERCQ, E
    AIDS RESEARCH AND HUMAN RETROVIRUSES, 1992, 8 (02) : 119 - 137
  • [36] OBSERVATIONS ON THE INHIBITION OF HIV-1 REVERSE-TRANSCRIPTASE BY CATECHINS
    MOORE, PS
    PIZZA, C
    BIOCHEMICAL JOURNAL, 1992, 288 : 717 - 719
  • [37] HIV-1 REVERSE-TRANSCRIPTASE EXPRESSION AND TRANSCOMPLEMENTATION ANALYSES
    ANSARILARI, MA
    DONEHOWER, LA
    GIBBS, RA
    JOURNAL OF CELLULAR BIOCHEMISTRY, 1995, : 185 - 185
  • [38] NEVIRAPINE BINDING DOMAIN FROM HIV-1 REVERSE-TRANSCRIPTASE CONFERS SENSITIVITY TO HIV-2 REVERSE-TRANSCRIPTASE
    BACOLLA, A
    HANSEN, GL
    ROSE, JM
    SHIH, CK
    GRIFFIN, JA
    FASEB JOURNAL, 1992, 6 (01): : A60 - A60
  • [39] Sexual transmission of an HIV-1 variant resistant to multiple reverse-transcriptase and protease inhibitors
    Hecht, FM
    Grant, RM
    Petropoulos, CJ
    Dillon, B
    Chesney, MA
    Tian, H
    Hellmann, NS
    Bandrapalli, NI
    Digilio, L
    Branson, B
    Kahn, JO
    NEW ENGLAND JOURNAL OF MEDICINE, 1998, 339 (05): : 307 - 311
  • [40] DEVELOPMENT OF A QUANTITATIVE IN-VITRO ASSAY TO STUDY INHIBITORS OF HIV-1 REVERSE-TRANSCRIPTASE
    KROGSTAD, P
    REY, O
    CANON, J
    JOURNAL OF CELLULAR BIOCHEMISTRY, 1995, : 193 - 193