SYNTHESIS AND PRELIMINARY EVALUATION OF TETRAHYDRONAPHTHALENE DERIVATIVES AS AMPA RECEPTOR ANTAGONISTS

被引：0
|
作者：
RETZ, DM [1 ]
BIGGE, CF [1 ]
RAFFERTY, MF [1 ]
机构：
[1] PARKE DAVIS PHARMACEUT RES DIV,ANN ARBOR,MI 48105
来源：
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 1994年 / 208卷
关键词：
D O I：
暂无
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
引用
收藏
页码：170 / MEDI
相关论文
共 50 条
  • [31] Synthesis and pharmacological evaluation of novel arylpiperazine derivatives as nonsteroidal androgen receptor antagonists
    Kinoyama, I
    Taniguchi, N
    Yoden, T
    Koutoku, H
    Furutani, T
    Kudoh, M
    Okada, M
    [J]. CHEMICAL & PHARMACEUTICAL BULLETIN, 2004, 52 (11) : 1330 - 1333
  • [32] Synthesis and pharmacological evaluation of coumarin derivatives as cannabinoid receptor antagonists and inverse agonists
    Behrenswerth, Andrea
    Volz, Nicole
    Toraeng, Jakob
    Hinz, Sonja
    Braese, Stefan
    Mueller, Christa E.
    [J]. BIOORGANIC & MEDICINAL CHEMISTRY, 2009, 17 (07) : 2842 - 2851
  • [33] SYNTHESIS AND EVALUATION OF NOVEL THIAZOLIDINE DERIVATIVES AS THROMBOXANE-A2 RECEPTOR ANTAGONISTS
    SATO, M
    KAWASHIMA, Y
    GOTO, J
    YAMANE, Y
    CHIBA, Y
    JINNO, S
    SATAKE, M
    IMANISHI, T
    IWATA, C
    [J]. CHEMICAL & PHARMACEUTICAL BULLETIN, 1994, 42 (03) : 521 - 529
  • [34] Design, Synthesis, and Preliminary Activity Evaluation of Novel Pyrimidine Derivatives as Acid Pump Antagonists
    Song, Weiguo
    Zhang, Xiaopan
    Li, Shutao
    Xu, Wenfang
    [J]. CHEMICAL BIOLOGY & DRUG DESIGN, 2015, 85 (03) : 306 - 314
  • [35] AMPA Receptor Antagonists for the Treatment of Stroke
    Weiser, Thomas
    [J]. CNS & NEUROLOGICAL DISORDERS-DRUG TARGETS, 2005, 4 (02) : 153 - 159
  • [36] Novel AMPA/kainate receptor antagonists
    Sakamoto, S
    Ohmori, J
    Shishikura, J
    ShimizuSasamata, M
    Okada, M
    [J]. MEDICINAL CHEMISTRY: TODAY AND TOMORROW, 1997, : 271 - 278
  • [37] Synthesis and preliminary pharmacological evaluation of a new putative radioiodinated AMPA receptor ligand for molecular imaging
    Ross, T. L.
    Sihver, W.
    Ermert, J.
    Coenen, H. H.
    [J]. RADIOCHIMICA ACTA, 2013, 101 (09) : 571 - 575
  • [38] Design and synthesis of novel quinoxaline-2,3-dione AMPA/GlyN receptor antagonists:: Amino acid derivatives
    Nikam, SS
    Cordon, JJ
    Ortwine, DF
    Heimbach, TH
    Blackburn, AC
    Vartanian, MG
    Nelson, CB
    Schwarz, RD
    Boxer, PA
    Rafferty, MF
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1999, 42 (12) : 2266 - 2271
  • [39] Synthesis and evaluation of diphenyl ether and decalin amino acids as AMPA antagonists
    Arnold, MB
    Ornstein, PL
    Allen, NK
    Schoepp, DD
    Wright, RA
    Johnson, DW
    Klimkowski, VJ
    [J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1996, 212 : 74 - MEDI
  • [40] NONPEPTIDIC ANGIOTENSIN-II ANTAGONISTS - SYNTHESIS AND INVITRO ACTIVITY OF A SERIES OF NOVEL NAPHTHALENE AND TETRAHYDRONAPHTHALENE DERIVATIVES
    BUHLMAYER, P
    CRISCIONE, L
    FUHRER, W
    FURET, P
    DEGASPARO, M
    STUTZ, S
    WHITEBREAD, S
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1991, 34 (10) : 3105 - 3114
12345