共 16 条
- [11] SINTEZ I PREVRASHCHENIE ALPHA-GLIKOLEI ETILENOVOGO RYADA .7. PREVRASHCHENIE 1,2,4-TRIFENILBUTEN-3-DIOLA-1,2 I 2,3-DIMETIL-5 FENILPENTEN-4-DIOLA-2,3 ZHURNAL OBSHCHEI KHIMII, 1959, 29 (07): : 2348 - 2354
- [14] Discovery of clinical candidate methyl (5-(6-((4(methylsulfonyl)piperazin-1-yl)methyl)-4-morpholinopyrrolo[2,1-f][1,2,4]triazin-2-yl)-4-(trifluoromethyl)pyridin-2-yl)carbamate (CYH33) : A highly potent and selective PI3K alpha inhibitor for the treatment of advanced solid tumors CANCER RESEARCH, 2018, 78 (13)
- [15] Identification of methyl (5-(6-((4-(methylsulfonyl)piperazin-1-yl)methyl)-4-morpholinopyrrolo[2,1-f][1,2,4]triazin-2-yl)-4-(trifluoromethyl)pyridin-2-yl)carbamate (CYH33) as an orally bioavailable, highly potent, PI3K alpha inhibitor for the treatment of advanced solid tumors EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 209
- [16] THE STRUCTURE AND ABSOLUTE-CONFIGURATION OF (22R)-3-BETA-ACETOXY-5-ALPHA,8-ALPHA-(3,5-DIOXO-4-PHENYL-1H,2H-1,2,4-TRIAZOLE-1,2-DIYL)-24-TRIMETHYLSILYLCHOL-6-EN-23-YN-22-YL P-BROMOBENZOATE AT 279 +/- 1 K ACTA CRYSTALLOGRAPHICA SECTION B-STRUCTURAL SCIENCE, 1980, 36 (OCT): : 2337 - 2341