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- [25] Discovery of ((1S,3R)-1-isopropyl-3-((3S,4S)-3-methoxy-tetrahydro-2H-pyran-4-ylamino)cyclopentyl)(4-(5-(trifluoromethyl)pyridazin-3-yl)piperazin-1-yl)methanone, PF-4254196, a CCR2 antagonist with an improved cardiovascular profile BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 21 (09) : 2626 - 2630
- [26] NEW SYNTHESIS OF 4,5-DIHYDRO-1,3-OXAZOLES AND 4,5-DIHYDRO-1,3-OXAZINES, USEFUL INTERMEDIATES TO ENANTIOMERICALLY PURE AMINO DIOLS - X-RAY MOLECULAR-STRUCTURE OF (4S,5R,4'S)-1-(4'-IODOMETHYL-4'-METHYL-4',5'-DIHYDRO-1',3'-OXAZOL-2'-YL)-3,4-DIMETHYL-5-PHENYLIMIDAZOLIDIN-2-ONE AND (4S,5R,4'S,1''S)-1-[4'-(1''-IODOBUTYL)-4',5'-DIHYDRO-1',3'-OXAZOL-2'-YL]-3,4-DIMETHYL-5-PHENYLIMIDAZOLIDIN-2-ONE JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 1990, (11): : 3095 - 3101
- [27] (1R,3S,6S)-6-tert-Butyl-1-hydroxymethyl-5-methoxy-6-methyl-7-oxa-4-azaspiro[2.5]oct-4-en-8-one and dimethyl[(1S,1R′,3S′,6S′)-(6′-tert-butyl-5′-methoxy-6′-methyl-8′-oxo-7′-oxa-4′-azaspiro[2.5]oct-4′-en-1′-yl)hydroxymethyl]phosphonate ACTA CRYSTALLOGRAPHICA SECTION C-STRUCTURAL CHEMISTRY, 2003, 59 : O317 - O320
- [28] (1S, 3aS, 4S, 7aS)-Ethyl1-benzyl-2-(4methoxybenzyl)-6,7-dimethyl-3-oxo-2,3,3a,4,5,7a-hexahydro-1H-isoindole4-carboxylate dichloromethane monosolvate ACTA CRYSTALLOGRAPHICA SECTION E-CRYSTALLOGRAPHIC COMMUNICATIONS, 2013, 69 : O316 - +
- [29] (3S,2′S,5′S,6′R,8′R,10′R)-3-hydroxy-4-(5′-hydroxy-10′-hydroxymethyl-5′-methyl-1′,7′,9′-trioxadispiro[5.1.5.2]pentadec-2′-yl)but-1-ene ACTA CRYSTALLOGRAPHICA SECTION E-CRYSTALLOGRAPHIC COMMUNICATIONS, 2006, 62 : O3968 - O3969