SYNTHESIS OF 1,2,3,4-TETRAHYDRO-5H-[1]BENZOPYRANO[3,4-C]PYRIDIN-5-ONES .2. SUBSTITUTION AT THE 3-POSITION WITH 2-AMINOETHYL AND 2-AMINOPROPYL SIDE-CHAINS

被引：9
|
作者：
CONNOR, DT
UNANGST, PC
SCHWENDER, CF
SORENSON, RJ
CARETHERS, ME
PUCHALSKI, C
BROWN, RE
机构：
来源：
JOURNAL OF HETEROCYCLIC CHEMISTRY | 1984年 / 21卷 / 05期
关键词：
D O I：
10.1002/jhet.5570210564
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Methods for the synthesis of 3-[2-aminoethyl]-1,2,3,4-tetrahydro-5H-[1]benzopyrano[3,4-c]pyridin-5-ones and 3-[2-aminopropyl]-1,2,3,4-tetrahydro-5H-[1]benzopyrano[3,4-c]pyridin-5-ones are described. The scope and limitations of the various methods are discussed. [These compounds could be useful in the treatment of asthma and bronchitis.].
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页码：1561 / 1564
页数：4
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