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- [41] Isolation and Identification of Three New 5-Alkenyl-3,3(2H)-furanones from Two Streptomyces species using a Genomic Screening ApproachThe Journal of Antibiotics, 2006, 59 : 168 - 176Arjun H Banskota论文数: 0 引用数: 0 h-index: 0机构: Ecopia BioSciences Inc.,James B McAlpine论文数: 0 引用数: 0 h-index: 0机构: Ecopia BioSciences Inc.,Dan Sørensen论文数: 0 引用数: 0 h-index: 0机构: Ecopia BioSciences Inc.,Mustapha Aouidate论文数: 0 引用数: 0 h-index: 0机构: Ecopia BioSciences Inc.,Mahmood Piraee论文数: 0 引用数: 0 h-index: 0机构: Ecopia BioSciences Inc.,Anne-Marie Alarco论文数: 0 引用数: 0 h-index: 0机构: Ecopia BioSciences Inc.,Satoshi Omura论文数: 0 引用数: 0 h-index: 0机构: Ecopia BioSciences Inc.,Kazuro Shiomi论文数: 0 引用数: 0 h-index: 0机构: Ecopia BioSciences Inc.,Chris M Farnet论文数: 0 引用数: 0 h-index: 0机构: Ecopia BioSciences Inc.,Emmanuel Zazopoulos论文数: 0 引用数: 0 h-index: 0机构: Ecopia BioSciences Inc.,
- [42] Optimization of Orally Bioavailable Enhancer of Zeste Homolog 2 (EZH2) Inhibitors Using Ligand and Property-Based Design Strategies: Identification of Development Candidate (R)-5,8-Dichloro-7-(methoxy(oxetan-3-yl)methyl)-2-((4-methoxy-6-methyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-3,4-dihydroisoquinolin-1(2H)-one (PF-06821497)JOURNAL OF MEDICINAL CHEMISTRY, 2018, 61 (03) : 650 - 665Kung, Pei-Pei论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USABingham, Patrick论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Res Unit, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USABrooun, Alexei论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USACollins, Michael论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USADeng, Ya-Li论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USADinh, Dac论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Res Unit, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USAFan, Connie论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Res Unit, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USAGajiwala, Ketan S.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USAGrantner, Rita论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Res Unit, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USAGukasyan, Hovhannes J.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Pharmaceut Sci Res Enabling Grp, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USAHu, Wenyue论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Drug Safety Res & Dev, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USAHuang, Buwen论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USAKania, Robert论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USAKephart, Susan E.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USAKrivacic, Cody论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Res Unit, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USAKumpf, Robert A.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USAKhamphavong, Penney论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Pharmaceut Sci Res Enabling Grp, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USAKraus, Manfred论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Res Unit, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USALiu, Wei论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USAMaegley, Karen A.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Res Unit, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USANguyen, Lisa论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Res Unit, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USARen, Shijian论文数: 0 引用数: 0 h-index: 0机构: WuXi AppTec, 288 Fute Zhong Rd, Shanghai 200131, Peoples R China Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USARichter, Dan论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USARollins, Robert A.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Res Unit, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, 401 N Middletown Rd, Pearl River, NY 10965 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USASach, Neal论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USASharma, Shikhar论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Res Unit, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USASherrill, John论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Res Unit, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USASpangler, Jillian论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USAStewart, Albert E.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USASutton, Scott论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USAUryu, Sean论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Res Unit, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USAVerhelle, Dominique论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Res Unit, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USAWang, Hui论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Res Unit, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USAWang, Shuiwang论文数: 0 引用数: 0 h-index: 0机构: WuXi AppTec, 288 Fute Zhong Rd, Shanghai 200131, Peoples R China Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USAWythes, Martin论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USAXin, Shuibo论文数: 0 引用数: 0 h-index: 0机构: WuXi AppTec, 288 Fute Zhong Rd, Shanghai 200131, Peoples R China Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USAYamazaki, Shinji论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Pharmacokinet Dynam & Metab, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USAZhu, Huichun论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USAZhu, JinJiang论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USAZehnder, Luke论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USAEdwards, Martin论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Global Res & Dev, La Jolla Labs, Oncol Med Chem, 10770 Sci Ctr Dr, San Diego, CA 92121 USA
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- [44] Synthesis of new 2-chloro-4-(3-aryl-2,4-diphenyl-3H-tria-zolidine-5-on-1-yl)quinoline-3-carbonitriles by a cycloaddition route using carbodiimides and nitrones. A novel thermal decomposition to 4-aminoquinolines.SYNTHETIC COMMUNICATIONS, 1998, 28 (19) : 3665 - 3674Mekheimer, RA论文数: 0 引用数: 0 h-index: 0机构: Menia Univ, Fac Sci, Dept Chem, Menia 61519, Egypt Menia Univ, Fac Sci, Dept Chem, Menia 61519, Egypt