HIGH-CAPACITY FOR PULMONARY 1ST-PASS ELIMINATION OF PROPRANOLOL IN RATS

被引:15
|
作者
IWAMOTO, K [1 ]
WATANABE, J [1 ]
AOYAMA, Y [1 ]
机构
[1] NAGOYA CITY UNIV,FAC PHARMACEUT SCI,DEPT BIOPHARMACEUT,NAGOYA,AICHI 467,JAPAN
关键词
D O I
10.1111/j.2042-7158.1987.tb03162.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:1049 / 1051
页数:3
相关论文
共 50 条
  • [1] AGE-DEPENDENT PULMONARY 1ST-PASS ELIMINATION OF PROPRANOLOL IN RATS
    IWAMOTO, K
    WATANABE, J
    AOYAMA, Y
    JOURNAL OF PHARMACY AND PHARMACOLOGY, 1988, 40 (02) : 135 - 137
  • [2] AVOIDANCE OF 1ST-PASS ELIMINATION OF RECTALLY ADMINISTERED PROPRANOLOL IN RELATION TO THE SITE OF ABSORPTION IN RATS
    DELEEDE, LGJ
    DEBOER, AG
    HAVERMANS, JPJM
    BREIMER, DD
    PHARMACEUTICAL RESEARCH, 1984, (04) : 164 - 168
  • [3] DOSE-DEPENDENT PRESYSTEMIC ELIMINATION OF PROPRANOLOL DUE TO HEPATIC 1ST-PASS METABOLISM IN RATS
    IWAMOTO, K
    WATANABE, J
    JOURNAL OF PHARMACY AND PHARMACOLOGY, 1985, 37 (11) : 826 - 828
  • [4] SATURABLE 1ST-PASS KINETICS OF PROPRANOLOL
    KELLER, F
    KUNZENDORF, U
    WALZ, G
    HALLER, H
    OFFERMANN, G
    JOURNAL OF CLINICAL PHARMACOLOGY, 1989, 29 (03): : 240 - 245
  • [5] EFFECT OF VITAMIN-K3 ON THE 1ST-PASS ELIMINATION OF PROPRANOLOL IN THE RAT
    ISHIDA, R
    USUI, T
    FUKUSHIMA, Y
    FUJITA, S
    SUZUKI, T
    JOURNAL OF PHARMACEUTICAL SCIENCES, 1985, 74 (05) : 578 - 581
  • [6] BIOAVAILABILITY AND PULMONARY 1ST-PASS REMOVAL OF ETRETINATE IN RATS
    THONGNOPNUA, P
    ZIMMERMAN, CL
    RESEARCH COMMUNICATIONS IN CHEMICAL PATHOLOGY AND PHARMACOLOGY, 1988, 61 (02): : 269 - 272
  • [7] NO STEREOSELECTIVE 1ST-PASS HEPATIC EXTRACTION OF PROPRANOLOL
    JACKMAN, GP
    MCLEAN, AJ
    JENNINGS, GL
    BOBIK, A
    CLINICAL PHARMACOLOGY & THERAPEUTICS, 1981, 30 (03) : 291 - 296
  • [8] GASTROINTESTINAL AND HEPATIC 1ST-PASS ELIMINATION OF 2',3'-DIDEOXYINOSINE IN RATS
    BRAMER, SL
    AU, JLS
    WIENTJES, MG
    JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 1993, 265 (02): : 731 - 738
  • [9] RECTAL BIOAVAILABILITY OF LIDOCAINE IN RATS - ABSENCE OF SIGNIFICANT 1ST-PASS ELIMINATION
    DEBOER, AG
    BREIMER, DD
    PRONK, J
    GUBBENSSTIBBE, JM
    JOURNAL OF PHARMACEUTICAL SCIENCES, 1980, 69 (07) : 804 - 807
  • [10] PARTIAL AVOIDANCE OF 1ST-PASS ELIMINATION OF AZATHIOPRINE IN RATS BY RECTAL DOSING
    TAKADA, K
    YOSHIKAWA, H
    MURANISHI, S
    INTERNATIONAL JOURNAL OF PHARMACEUTICS, 1985, 25 (02) : 155 - 163