2-DIBENZYLAMINOBUTANE-1,4-DIOL - A VERSATILE INTERMEDIATE FOR A CHIROSPECIFIC BETA-AMINO ACID SYNTHESIS

被引：23

作者：

GMEINER, P

ORECHER, F

THOMAS, C

WEBER, K

机构：

[1] Pharmazeutisches Institut der Universität Bonn, D-53121 Bonn

来源：

TETRAHEDRON LETTERS | 1995年 / 36卷 / 03期

关键词：

D O I：

10.1016/0040-4039(94)02307-W

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Starting from the chiral building block 1, which is readily available from natural aspartic acid, a concise and versatile synthesis of optically active beta-amino acids including beta-proline derivatives is reported. Regioselective transformations of the 1,4-bis-electrophile 2 are facilitated by an anchimeric participation.

引用

页码：381 / 382

页数：2

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