PREPARATION OF 2,2-DISUBSTITUTED 2,3-DIHYDRO-3-PHENYL-1,3,4-THIADIAZOLES

被引：0
|
作者：
KITANO, K [1 ]
MATSUBARA, Y [1 ]
YOSHIHARA, M [1 ]
MAESHIMA, T [1 ]
机构：
[1] KINKI UNIV, FAC SCI & ENGN, DEPT APPL CHEM, OSAKA 577, JAPAN
来源：
CHEMICAL & PHARMACEUTICAL BULLETIN | 1994年 / 42卷 / 09期
关键词：
2,3-DIHYDRO-3-PHENYL-1,3,4-THIADIAZOLE; TRIMETHYLSILYL CHLORIDE; KETONE; CYCLIZATION;
D O I：
暂无
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
Reaction of N'-phenylthioformohydrazide with ketones in the presence of trimethylsilyl chloride proceeded easily to afford the corresponding 2,2-disubstituted 2,3-dihydro-3-phenyl-1,3,4-thiadiazoles in good yields.
引用
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页码：1912 / 1913
页数：2
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