PREPARATION OF 2,2-DISUBSTITUTED 2,3-DIHYDRO-3-PHENYL-1,3,4-THIADIAZOLES

被引：0

作者：

KITANO, K ^{[1
]}

MATSUBARA, Y ^{[1
]}

YOSHIHARA, M ^{[1
]}

MAESHIMA, T ^{[1
]}

机构：

[1] KINKI UNIV, FAC SCI & ENGN, DEPT APPL CHEM, OSAKA 577, JAPAN

来源：

CHEMICAL & PHARMACEUTICAL BULLETIN | 1994年 / 42卷 / 09期

关键词：

2,3-DIHYDRO-3-PHENYL-1,3,4-THIADIAZOLE; TRIMETHYLSILYL CHLORIDE; KETONE; CYCLIZATION;

D O I：

暂无

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

Reaction of N'-phenylthioformohydrazide with ketones in the presence of trimethylsilyl chloride proceeded easily to afford the corresponding 2,2-disubstituted 2,3-dihydro-3-phenyl-1,3,4-thiadiazoles in good yields.

引用

页码：1912 / 1913

页数：2

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