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- [44] Mechanistic Study of Potent Fluorinated EGFR Kinase Inhibitors with a Quinazoline Scaffold against L858R/T790M/C797S Resistance Mutation: Unveiling the Fluorine Substituent Cooperativity Effect on the Inhibitory Activity JOURNAL OF PHYSICAL CHEMISTRY B, 2020, 124 (28): : 5813 - 5824