DISPOSITION OF ENALAPRIL IN THE PERFUSED RAT INTESTINE-LIVER PREPARATION - ABSORPTION, METABOLISM AND 1ST-PASS EFFECT

被引:0
|
作者
PANG, KS [1 ]
CHERRY, WF [1 ]
ULM, EH [1 ]
机构
[1] MERCK SHARP & DOHME RES LABS,MERCK INST THERAPEUT RES,W POINT,PA 19486
关键词
D O I
暂无
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:788 / 795
页数:8
相关论文
共 50 条
  • [31] ORAL ABSORPTION AND PRESYSTEMIC 1ST-PASS EFFECT OF CHLORPHENIRAMINE IN RABBITS
    HUANG, SM
    HUANG, YC
    CHIOU, WL
    [J]. JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS, 1981, 9 (06): : 725 - 738
  • [32] INFLUENCE OF DOSE ON 1ST-PASS KINETICS OF IMIPRAMINE-C-14 IN THE ISOLATED PERFUSED RAT-LIVER
    BEAUBIEN, AR
    PAKUTS, AP
    [J]. DRUG METABOLISM AND DISPOSITION, 1979, 7 (01) : 34 - 39
  • [33] SEX-DIFFERENCES IN 1ST-PASS EXTRACTION OF INDOCYANINE GREEN (ICG) IN THE ISOLATED PERFUSED RAT-LIVER
    KUSHLAN, M
    GOLLAN, J
    MA, WL
    OCKNER, R
    [J]. GASTROENTEROLOGY, 1979, 77 (05) : A23 - A23
  • [34] NONLINEAR BIOAVAILABILITY OF METOCLOPRAMIDE IN THE RAT - EVIDENCE FOR SATURABLE 1ST-PASS METABOLISM
    KAPIL, RP
    AXELSON, JE
    ONGLEY, R
    PRICE, JDE
    [J]. JOURNAL OF PHARMACEUTICAL SCIENCES, 1984, 73 (02) : 215 - 218
  • [35] 1ST-PASS GASTRIC-MUCOSAL METABOLISM OF ETHANOL IS NEGLIGIBLE IN THE RAT
    SMITH, T
    DEMASTER, EG
    FURNE, JK
    SPRINGFIELD, J
    LEVITT, MD
    [J]. JOURNAL OF CLINICAL INVESTIGATION, 1992, 89 (06): : 1801 - 1806
  • [36] DISPOSITION OF LORAZEPAM IN HUMAN-BEINGS - ENTEROHEPATIC RECIRCULATION AND 1ST-PASS EFFECT
    HERMAN, RJ
    VANPHAM, JD
    SZAKACS, CBN
    [J]. CLINICAL PHARMACOLOGY & THERAPEUTICS, 1989, 46 (01) : 18 - 25
  • [37] ABSORPTION AND METABOLISM OF ACETAMINOPHEN BY THE INSITU PERFUSED RAT SMALL-INTESTINE PREPARATION
    PANG, KS
    YUEN, V
    FAYZ, S
    TEKOPPELE, JM
    MULDER, GJ
    [J]. DRUG METABOLISM AND DISPOSITION, 1986, 14 (01) : 102 - 111
  • [38] ABSORPTION AND 1ST-PASS METABOLISM OF GAMMA-HYDROXYBUTYRIC-C-14 ACID
    LETTIERI, J
    FUNG, HL
    [J]. RESEARCH COMMUNICATIONS IN CHEMICAL PATHOLOGY AND PHARMACOLOGY, 1976, 13 (03): : 425 - 437
  • [39] EFFECT OF GLIBENCLAMIDE ON THE ABSORPTION AND METABOLISM OF GLUCOSE BY THE INVITRO PERFUSED RAT INTESTINE
    ZUBELDIA, MAG
    TORMO, MA
    MONTERO, JL
    ROPERO, MF
    CAMPILLO, JE
    [J]. DIABETES NUTRITION & METABOLISM, 1993, 6 (02) : 67 - 70
  • [40] INTESTINAL 1ST-PASS METABOLISM OF NITROSAMINES .2. METABOLISM OF N-NITROSODIBUTYLAMINE IN ISOLATED PERFUSED RAT SMALL INTESTINAL SEGMENTS
    RICHTER, E
    ZWICKENPFLUG, W
    WIESSLER, M
    [J]. CARCINOGENESIS, 1988, 9 (03) : 499 - 506