DIFFERENTIAL INTERACTION OF THE OPIOID RECEPTOR WITH AGONIST AND ANTAGONIST MORPHINAN DERIVATIVES

被引:0
|
作者
LEMAIRE, S
BELLEAU, B
机构
[1] UNIV OTTAWA, FAC HLTH SCI, DEPT PHARMACOL, OTTAWA K1N 6N5, ONTARIO, CANADA
[2] MCGILL UNIV, DEPT CHEM, MONTREAL H3A 2T5, QUEBEC, CANADA
来源
FASEB JOURNAL | 1988年 / 2卷 / 05期
关键词
D O I
暂无
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:A1391 / A1391
页数:1
相关论文
共 50 条
  • [41] Differential effects of LY235959, a competitive antagonist of the NMDA receptor on kappa-opioid receptor agonist induced responses in mice and rats
    Bhargava, HN
    Thorat, SN
    BRAIN RESEARCH, 1997, 747 (02) : 246 - 251
  • [42] RECEPTOR ANTAGONIST AND SELECTIVE AGONIST DERIVATIVES OF MOUSE INTERLEUKIN-2
    ZURAWSKI, SM
    ZURAWSKI, G
    EMBO JOURNAL, 1992, 11 (11): : 3905 - 3910
  • [43] In vivo antinociception of potent mu opioid agonist tetrapeptide analogues and comparison with a compact opioid agonist - neurokinin 1 receptor antagonist chimera
    Guillemyn, Karel
    Kleczkowska, Patrycja
    Novoa, Alexandre
    Vandormael, Bart
    Van den Eynde, Isabelle
    Kosson, Piotr
    Asim, Muhammad Faheem
    Schiller, Peter W.
    Spetea, Mariana
    Lipkowski, Andrzej W.
    Tourwe, Dirk
    Ballet, Steven
    MOLECULAR BRAIN, 2012, 5
  • [44] In vivo antinociception of potent mu opioid agonist tetrapeptide analogues and comparison with a compact opioid agonist - neurokinin 1 receptor antagonist chimera
    Karel Guillemyn
    Patrycja Kleczkowska
    Alexandre Novoa
    Bart Vandormael
    Isabelle Van den Eynde
    Piotr Kosson
    Muhammad Faheem Asim
    Peter W Schiller
    Mariana Spetea
    Andrzej W Lipkowski
    Dirk Tourwé
    Steven Ballet
    Molecular Brain, 5
  • [45] Syntheses and receptor-binding studies of derivatives of the opioid antagonist naltrexone
    Uwai, K
    Uchiyama, H
    Sakurada, S
    Kabuto, C
    Takeshita, M
    BIOORGANIC & MEDICINAL CHEMISTRY, 2004, 12 (02) : 417 - 421
  • [46] New therapeutic options for IBS: the role of the first in class mixed μ-opioid receptor agonist and δ-opioid receptor antagonist (mudelta) eluxadoline
    Corsetti, Maura
    Whorwell, Peter
    EXPERT REVIEW OF GASTROENTEROLOGY & HEPATOLOGY, 2017, 11 (04) : 285 - 292
  • [48] Peptidomimetics Exhibiting Mu Opioid Receptor (MOPr) Agonist/Delta Opioid Receptor (DOPr) Antagonist Activity as Novel Pain Therapeutics
    Griggs, Nicholas
    Bender, Aaron
    Gao, Chao
    Anand, Jessica
    Traynor, John
    Mosberg, Henry
    FASEB JOURNAL, 2016, 30
  • [49] THERMODYNAMICS OF AGONIST AND ANTAGONIST INTERACTION WITH THE STRYCHNINE-SENSITIVE GLYCINE RECEPTOR
    RUIZGOMEZ, A
    GARCIACALVO, M
    VAZQUEZ, J
    MARVIZON, JCG
    VALDIVIESO, F
    MAYOR, F
    JOURNAL OF NEUROCHEMISTRY, 1989, 52 (06) : 1775 - 1780
  • [50] Differential time course of effects of κ-opioid agonist treatment on dynorphin a levels and κ-opioid receptor density
    Claudio D’Addario
    Manuela Di Benedetto
    Sari Izenwasser
    Sanzio Candeletti
    Patrizia Romualdi
    Journal of Molecular Neuroscience, 2004, 24 : 307 - 314