SYNTHESIS OF FUNCTIONALIZED INDOLES BY DIELS-ALDER REACTION UTILIZING THE DIENE GENERATED BY THE ALKYLATION OF N-METHYL-3-THIOACETYLPYRROLE

被引：0

作者：

MURASE, M ^{[1
]}

YOSHIDA, S ^{[1
]}

HOSAKA, T ^{[1
]}

TOBINAGA, S ^{[1
]}

机构：

[1] SHOWA COLL PHARMACEUT SCI, TOKYO 194, JAPAN

来源：

CHEMICAL & PHARMACEUTICAL BULLETIN | 1991年 / 39卷 / 02期

关键词：

CYCLOADDITION; 3-VINYLPYRROLE; 1-METHYL-3-THIOACETYLPYRROLE; ALKYLATION; DIENOPHILE; INDOLE;

D O I：

暂无

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

Cycloaddition reaction of 3-vinylpyrroles, generated by the alkylation of 1-methyl-3-thioacetylpyrrole, with dienophiles provided functionalized indoles.

引用

页码：489 / 492

页数：4

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