Synthesis and antifungal activity of 3-substituted thiochromanones

被引：2
|
作者：
Liu, Yang [1 ]
Luo, Wei [1 ]
Sun, Li [1 ]
Guo, Chun [1 ]
机构：
[1] Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Shenyang, Liaoning, Peoples R China
来源：
DRUG DISCOVERIES AND THERAPEUTICS | 2008年 / 2卷 / 04期
关键词：
Thiochromanone; Synthesis; Antifungal activity;
D O I：
暂无
中图分类号：
R9 [药学];
学科分类号：
1007 ;
摘要：
A series of 3-substituted thiochromanones has been prepared. Their structures were confirmed by H-1-NMR and HRMS. All of the synthesized compounds were screened for antifungal activity against ten fungi species in vitro. The compounds 2f and 2g were more efficient than the control drug, ketoconazole.
引用
收藏
页码：216 / 218
页数：3
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