Convenient Synthetic Approach to (2-Aryl-5-phenyl-1,3-oxazol-4-yl)phosphonic Acids and Their Functional Derivatives

被引:0
|
作者
A. G. Belyuga
V. S. Brovarets
B. S. Drach
机构
[1] National Academy of Sciences of Ukraine,Institute of Bioorganic Chemistry and Petrochemistry
来源
关键词
Phosphorus; Successive Treatment; General Formula; Trimethyl; Phosphite;
D O I
暂无
中图分类号
学科分类号
摘要
Successive treatment of available amidophenacylating agents of the general formula PhCOCH ⋅ ClNHCOAr with trimethyl phosphite and phosphorus pentachloride gave previously unknown (2-aryl-5-phenyl-1,3-oxazol-4-yl)phosphonic dichlorides which are suitable dtarting materials for preparing other phosphorylated oxazoles containing P(O)(OH)2, P(O)(NHAlk)2, P(O)(OMe)NHAlk, P(O)(OMe)NAlk2, and other groups in the 4 position of the heteroring.
引用
收藏
页码:523 / 526
页数:3
相关论文
共 50 条
  • [21] (4Z)-4-Benzylidene-2-phenyl-1,3-oxazol-5-(4H)-one
    Asiri, Abdullah M.
    Faidallah, Hassan M.
    Sobahi, Tariq R.
    Ng, Seik Weng
    Tiekink, Edward R. T.
    ACTA CRYSTALLOGRAPHICA SECTION E-CRYSTALLOGRAPHIC COMMUNICATIONS, 2015, 71 : E4 - E4
  • [22] NEW SYNTHETIC PYRETHROIDS - 4-PHENYL-2-BUTEN-1-YL AND 4-ARYL-2-BUTYN-1-YL CHRYSANTHEMATES
    SOTA, K
    AMANO, T
    AIDA, M
    NODA, K
    HAYASHI, A
    TANAKA, I
    AGRICULTURAL AND BIOLOGICAL CHEMISTRY, 1971, 35 (06): : 968 - &
  • [23] 2,6-dimethoxy-4-(5-oxo-2-phenyl-4,5-dihydro-1,3-oxazol-4-ylidenemethyl)-phenyl acetate
    Sun, Yi-Feng
    Wang, Xin-Li
    Li, Ji-Kun
    Zheng, Ze-Bao
    Wu, Ren-Tao
    ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE, 2007, 63 : O4426 - U4415
  • [24] Reaction of 2-aryl-4-dichloromethylidene-1,3-oxazol-5(4H)-ones with 2-aminopyridine
    Prokopenko, V. M.
    Pil'o, S. G.
    Brovarets, V. S.
    Vasilenko, A. N.
    Drach, B. S.
    RUSSIAN JOURNAL OF GENERAL CHEMISTRY, 2010, 80 (01) : 121 - 126
  • [25] Reaction of 2-aryl-4-dichloromethylidene-1,3-oxazol-5(4H)-ones with 2-aminopyridine
    V. M. Prokopenko
    S. G. Pil’o
    V. S. Brovarets
    A. N. Vasilenko
    B. S. Drach
    Russian Journal of General Chemistry, 2010, 80 : 121 - 126
  • [26] A convenient method for the synthesis of 2-[(5-benzyl-1,3-thiazol-2-yl)imino]-1,3-thiazolidin-4-one derivatives
    Ostapiuk, Yuri V.
    Obushak, Mykola D.
    Matiychuk, Vasyl S.
    Naskrent, Marek
    Gzella, Andrzej K.
    TETRAHEDRON LETTERS, 2012, 53 (05) : 543 - 545
  • [27] Synthesis, Antibacterial, and Antimonooxidase Activity of 4-(2-Methyl-1,3-oxazol-5-yl)benzenesulfonamide
    Gasilina, O. A.
    Romanycheva, A. A.
    Shetnev, A. A.
    Korsakov, M. K.
    RUSSIAN JOURNAL OF GENERAL CHEMISTRY, 2023, 93 (11) : 2749 - 2755
  • [28] Synthesis, Antibacterial, and Antimonooxidase Activity of 4-(2-Methyl-1,3-oxazol-5-yl)benzenesulfonamide
    O. A. Gasilina
    A. A. Romanycheva
    A. A. Shetnev
    M. K. Korsakov
    Russian Journal of General Chemistry, 2023, 93 : 2749 - 2755
  • [29] 2-Methoxy-4-[(5-oxo-2-phenyl-4,5-dihydro-1,3-oxazol-4-ylidene)methyl]-phenyl 4-methylbenzenesulfonate
    Sen, Betul
    Ozturk, Gulsiye
    Alp, Serap
    Aygun, Muhittin
    Buyukgungor, Orhan
    ACTA CRYSTALLOGRAPHICA SECTION C-CRYSTAL STRUCTURE COMMUNICATIONS, 2007, 63 : O223 - O224
  • [30] SYNTHESIS AND REACTIONS OF 5-BENZYLIDENE-2-PHENYL-4,5-DIHYDRO-1,3-OXAZOL-4-ONES
    LAXMI, YS
    IYENGAR, DS
    JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 1995, (23): : 3043 - 3045