Convenient Synthetic Approach to (2-Aryl-5-phenyl-1,3-oxazol-4-yl)phosphonic Acids and Their Functional Derivatives

被引：0
|
作者：
A. G. Belyuga
V. S. Brovarets
B. S. Drach
机构：
[1] National Academy of Sciences of Ukraine,Institute of Bioorganic Chemistry and Petrochemistry
来源：
Russian Journal of General Chemistry | 2005年 / 75卷
关键词：
Phosphorus; Successive Treatment; General Formula; Trimethyl; Phosphite;
D O I：
暂无
中图分类号：
学科分类号：
摘要：
Successive treatment of available amidophenacylating agents of the general formula PhCOCH ⋅ ClNHCOAr with trimethyl phosphite and phosphorus pentachloride gave previously unknown (2-aryl-5-phenyl-1,3-oxazol-4-yl)phosphonic dichlorides which are suitable dtarting materials for preparing other phosphorylated oxazoles containing P(O)(OH)2, P(O)(NHAlk)2, P(O)(OMe)NHAlk, P(O)(OMe)NAlk2, and other groups in the 4 position of the heteroring.
引用
收藏
页码：523 / 526
页数：3
相关论文
共 50 条
  • [1] Convenient synthetic approach to (2-aryl-5-phenyl-1,3-oxazol-4-yl)phosphonic acids and their functional derivatives
    Belyuga, AG
    Brovarets, VS
    Drach, BS
    RUSSIAN JOURNAL OF GENERAL CHEMISTRY, 2005, 75 (04) : 523 - 526
  • [2] Synthesis and properties of methanesulfonyl derivatives of diethyl esters of 5-(hydroxyalkylamino)-1,3-oxazol-4-yl-phosphonic acids
    Golovchenko, O. V.
    Brusnakov, M. Yu.
    Shabelko, Yu. O.
    Brovarets, V. S.
    Vydzhak, R. M.
    Bahrieieva, O. S.
    Potikha, L. M.
    Shishkina, S. V.
    PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS, 2024, 199 (01) : 71 - 81
  • [3] 2-[(2-Phenyl-1,3-oxazol-4-yl)methyl]-2H-1,2,3-benzo-triazole
    Swaleh, S
    Ziemer, B
    ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE, 2001, 57 : O35 - O36
  • [4] 4-ARYLBUTADIEN-1,3-YL PHOSPHONIC ACIDS AND THEIR DERIVATIVES
    GANUSHCHAK, NI
    FEDOROVA, GK
    VENGRZHA.VA
    ZHURNAL OBSHCHEI KHIMII, 1972, 42 (02): : 291 - +
  • [5] Synthesis and spectral properties of 3-(2-aryl-5-methyl-1,3-oxazol-4-yl)-2-(2,5-dimethylthiophen-3-yl)cyclopent-2-en-1-ones
    Lvov, Andrey G.
    Shirinian, Valerii Z.
    Kavun, Alexey M.
    Krayushkin, Mikhail M.
    MENDELEEV COMMUNICATIONS, 2014, 24 (05) : 277 - 279
  • [6] 5-(4-Fluorophenyl)-2-[2-(5-phenyl-1,3-oxazol-2-yl)phenyl]-1,3-oxazole
    Ilyashenko, Rodion
    Wera, Michal
    Blazejowski, Jerzy
    Doroshenko, Andrey
    ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE, 2010, 66 : O2379 - U919
  • [7] Synthesis of 2-methoxy-2-methyl-3-{6-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]pyridin-3-yl}propanoic acid, a dual PPARα/γ agonist
    Humphries, Paul S.
    Do, Quyen-Quyen T.
    Wilhite, David M.
    TETRAHEDRON LETTERS, 2009, 50 (16) : 1765 - 1767
  • [8] Structural characterization of new 2-aryl-5-phenyl-1,3, 4-oxadiazin-6-ones and their N-aroylhydrazone precursors
    Tintas, Mihaela Liliana
    Diac, Andreea Petronela
    Soran, Albert
    Terec, Anamaria
    Grosu, Ion
    Bogdan, Elena
    JOURNAL OF MOLECULAR STRUCTURE, 2014, 1058 : 106 - 113
  • [9] 4-chloro-2-{4-[p-(methylsulfonyl)phenyl]-2-oxo-5-phenyl-2,3-dihydro-1,3-oxazol-3-yl}-phenyl acetate
    Tsou, NN
    Ball, RG
    Roy, PJ
    Leblanc, Y
    ACTA CRYSTALLOGRAPHICA SECTION C-CRYSTAL STRUCTURE COMMUNICATIONS, 1998, 54 : 1493 - 1494
  • [10] Antileshmanial Activities of Synthetic Substituted 2-phenyl-4-[phenylmethylidene]-1,3-oxazol-5(4H)-ones
    Khan, Saadia Razi
    Ghouri, Nida
    Karim, Aneela
    Naz, Farzana
    Fakhri, Muhammad Imran
    Perveen, Shahnaz
    Khan, Khalid Mohammed
    Taha, Muhammad
    Choudhary, Muhammad Iqbal
    JOURNAL OF THE CHEMICAL SOCIETY OF PAKISTAN, 2015, 37 (05): : 980 - 985
12345