Synthesis of stereoisomeric 4-(2-methylindolin-1-yl)- and 4-(2-methylindol-1-yl) derivatives of glutamic acid

被引：0
|
作者：
V. P. Krasnov
A. Yu. Vigorov
I. A. Nizova
A. N. Grishakov
N. G. Evstigneeva
M. I. Kodess
机构：
[1] Ural Branch of the Russian Academy of Sciences,I. Ya. Postovsky Institute of Organic Synthesis
来源：
Russian Chemical Bulletin | 2004年 / 53卷
关键词：
glutamic acid; 2-methylindoline; 2-methylindole; nucleophilic substitution; stereoisomers;
D O I：
暂无
中图分类号：
学科分类号：
摘要：
The reaction of dimethyl (2S,4RS)-N-phthaloyl-4-bromoglutamate with 2-methylindoline afforded diastereomeric 4-(2-methylindolin-1-yl)-(S)-glutamic acid derivatives, whose oxidation gave rise to 4-(2-methylindol-1-yl)-(S)-glutamic acid derivatives.
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收藏
页码：1327 / 1330
页数：3
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