[18F]F15599, a novel 5-HT1A receptor agonist, as a radioligand for PET neuroimaging

被引:0
|
作者
Laëtitia Lemoine
Mathieu Verdurand
Bernard Vacher
Elodie Blanc
Didier Le Bars
Adrian Newman-Tancredi
Luc Zimmer
机构
[1] Université de Lyon,Laboratory of Neuropharmacology
[2] CERMEP – Imagerie du Vivant,PET Department
[3] CERMEP – Imagerie du Vivant,ANIMAGE Department
[4] Centre de Recherches Pierre Fabre,undefined
关键词
Serotonin 1A receptor; PET; Agonist; Rat; Cat;
D O I
暂无
中图分类号
学科分类号
摘要
引用
收藏
页码:594 / 605
页数:11
相关论文
共 50 条
  • [31] F15599, a post-synaptic cortical preferential 5-HT1A agonist: II) Effect in rodent models of cognition/memory deficits
    Depoortere, R.
    Auclair, A.
    Bardin, L.
    Newman-Tancredi, A.
    EUROPEAN NEUROPSYCHOPHARMACOLOGY, 2008, 18 : S353 - S353
  • [32] F15599, a post-synaptic cortical preferential 5-HT1A agonist: I) functionally-selective signal transduction profile
    Newman-Tancredi, A.
    Martel, J. C.
    Buritova, J.
    Lauressergues, E.
    Assie, M. B.
    Slot, L. Bruins
    Cosi, C.
    Heusler, P.
    Cussac, D.
    EUROPEAN NEUROPSYCHOPHARMACOLOGY, 2008, 18 : S352 - S353
  • [33] Aggression-reducing effects of F15599, a novel selective 5-HT1A receptor agonist, after microinjection into the ventral orbital prefrontal cortex, but not in infralimbic cortex in male mice
    Dirson João Stein
    Klaus A. Miczek
    Aldo Bolten Lucion
    Rosa Maria Martins de Almeida
    Psychopharmacology, 2013, 230 : 375 - 387
  • [34] F15599, a highly selective serotonin 5-HT1A receptor agonist that preferentially targets post-synaptic receptors in the frontal cortex:: biochemical and neurochemical profiles
    Auclair, A.
    Buritova, Y.
    Cussac, D.
    Assie, M-B
    Depoortere, R.
    Newman-Tancredi, A.
    FUNDAMENTAL & CLINICAL PHARMACOLOGY, 2008, 22 : 117 - 117
  • [35] PET evaluation of [18F]FCWAY, an analog of the 5-HT1A receptor antagonist, WAY-100635
    Carson, RE
    Lan, LX
    Watabe, H
    Der, MG
    Adams, HR
    Jagoda, E
    Herscovitch, P
    Eckelman, WC
    NUCLEAR MEDICINE AND BIOLOGY, 2000, 27 (05) : 493 - 497
  • [36] p-[18F]-MPPF PET imaging of 5-HT1A receptor binding in marmoset brain
    Converse, Alexander K.
    Aubert, Y.
    Murali, D.
    Weichert, J. P.
    DeJesus, O. T.
    Nickles, R. J.
    Abbott, D. H.
    NEUROIMAGE, 2008, 41 : T148 - T148
  • [37] [18F]Mefway PET imaging of serotonin 5-HT1A receptors in hu ans
    Hillmer, Ansel
    Wooten, Dustin
    Lao, Patrick
    Betthauser, Tobey
    Barnhart, Todd
    Rowley, Howard
    Hall, Lance
    Stone, Charles
    Mukherjee, Jogeshwar
    Christian, Bradley
    JOURNAL OF NUCLEAR MEDICINE, 2014, 55
  • [38] [18F]F13640, a 5-HT1A Receptor Radiopharmaceutical Sensitive to Brain Serotonin Fluctuations
    Colom, Matthieu
    Vidal, Benjamin
    Fieux, Sylvain
    Redoute, Jerome
    Costes, Nicolas
    Lavenne, Franck
    Merida, Ines
    Irace, Zacharie
    Iecker, Thibaud
    Bouillot, Caroline
    Billard, Thierry
    Newman-Tancredi, Adrian
    Zimmer, Luc
    FRONTIERS IN NEUROSCIENCE, 2021, 15
  • [39] The effects of a total sleep deprivation on the brain 5-HT1A receptor binding:: A pet study with [18F]MPPF
    Lakhdarchaouche, Y
    Faivre, T
    Costes, N
    Zimmer, L
    Nicolas, A
    Fort, P
    Lemoine, P
    Luppi, P
    INTERNATIONAL JOURNAL OF NEUROPSYCHOPHARMACOLOGY, 2004, 7 : S286 - S286
  • [40] 5-HT1A binding of [18F]MEFWAY in the rhesus monkey
    Wooten, Dustin
    Hillmer, Ansel
    Moirano, Jeffrey
    Tudorascu, Dana
    Murali, Dhanabalan
    Barnhart, Todd
    Kallin, Ned
    Davidson, Richard
    Mukherjee, Jogesh
    Schneider, Mary
    Christian, Brad
    NEUROIMAGE, 2010, 52 : S129 - S130